← Mechanisms of action
GABA-B receptor
PROTEIN COMPLEXHomo sapiens
Linked proteins
Drugs acting on this target (4)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| arbaclofen | Agonist | experimental | Small molecule | GABA-B receptor agonist |
| baclofen (lioresal) | Agonist | approved | Small molecule | GABA-B receptor agonist |
| sodium oxybate (xyrem) | Agonist | approved | Small molecule | GABA-B receptor agonist |
| sgs-742 | Antagonist | experimental | Small molecule | GABA-B receptor antagonist |