← Mechanisms of action

GABBR1

SINGLE PROTEINHomo sapiens
Preferred name: GABA-B receptor 1 ChEMBL ↗

Linked proteins

Drugs acting on this target (6)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
odm-106ActivatorexperimentalSmall moleculeGABBR1 activator
lesogaberanAgonistexperimentalSmall moleculeGABBR1 agonist
ValiloxybateAgonistexperimentalSmall moleculeGABBR1 agonist
bd114Allosteric antagonistexperimentalSmall moleculeGABBR1 allosteric antagonist
sgs-742AntagonistexperimentalSmall moleculeGABBR1 antagonist
asp8062InhibitorexperimentalSmall moleculeGABBR1 inhibitor