← Mechanisms of action
Rho-associated protein kinase
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (11)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ama-0076 | Inhibitor | experimental | Small molecule | Rho-associated protein kinase inhibitor |
| at13148 | Inhibitor | experimental | Small molecule | Rho-associated protein kinase inhibitor |
| belumosudil (Rezurock) | Inhibitor | approved | Small molecule | Rho-associated protein kinase inhibitor |
| de-104 | Inhibitor | experimental | Small molecule | Rho-associated protein kinase inhibitor |
| fasudil | Inhibitor | experimental | Small molecule | Rho-associated protein kinase inhibitor |
| k-321 | Inhibitor | experimental | Small molecule | Rho-associated protein kinase inhibitor |
| netarsudil (Rhopressa) | Inhibitor | approved | Small molecule | Rho-associated protein kinase inhibitor |
| ripasudil (Glanatec) | Inhibitor | experimental | Small molecule | Rho-associated protein kinase inhibitor |
| sar-407899 | Inhibitor | experimental | Small molecule | Rho-associated protein kinase inhibitor |
| verosudil | Inhibitor | experimental | Small molecule | Rho-associated protein kinase inhibitor |
| y-39983 | Inhibitor | experimental | Small molecule | Rho-associated protein kinase inhibitor |