← Mechanisms of action

Rho-associated protein kinase

PROTEIN FAMILYHomo sapiens

Linked proteins

Drugs acting on this target (11)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
ama-0076InhibitorexperimentalSmall moleculeRho-associated protein kinase inhibitor
at13148InhibitorexperimentalSmall moleculeRho-associated protein kinase inhibitor
belumosudil (Rezurock)InhibitorapprovedSmall moleculeRho-associated protein kinase inhibitor
de-104InhibitorexperimentalSmall moleculeRho-associated protein kinase inhibitor
fasudilInhibitorexperimentalSmall moleculeRho-associated protein kinase inhibitor
k-321InhibitorexperimentalSmall moleculeRho-associated protein kinase inhibitor
netarsudil (Rhopressa)InhibitorapprovedSmall moleculeRho-associated protein kinase inhibitor
ripasudil (Glanatec)InhibitorexperimentalSmall moleculeRho-associated protein kinase inhibitor
sar-407899InhibitorexperimentalSmall moleculeRho-associated protein kinase inhibitor
verosudilInhibitorexperimentalSmall moleculeRho-associated protein kinase inhibitor
y-39983InhibitorexperimentalSmall moleculeRho-associated protein kinase inhibitor