← Mechanisms of action
ROCK2
SINGLE PROTEINHomo sapiens
Preferred name: Rho-associated protein kinase 2 ChEMBL ↗
Linked proteins
Drugs acting on this target (14)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| belumosudil (Rezurock) | Antagonist | approved | Small molecule | ROCK2 antagonist |
| AR-13154 | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| ats907 | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| belumosudil (Rezurock) | Inhibitor | approved | Small molecule | Rho-associated protein kinase 2 inhibitor |
| cethrin | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| fasudil | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| gns-3545 | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| gv101 | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| opl-0401 | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| ripasudil (Glanatec) | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| roc-101 | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| tdi01 | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| tq05105 | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |
| Zelasudil | Inhibitor | experimental | Small molecule | ROCK2 inhibitor |