← Mechanisms of action

ROCK2

SINGLE PROTEINHomo sapiens
Preferred name: Rho-associated protein kinase 2 ChEMBL ↗

Linked proteins

Drugs acting on this target (14)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
belumosudil (Rezurock)AntagonistapprovedSmall moleculeROCK2 antagonist
AR-13154InhibitorexperimentalSmall moleculeROCK2 inhibitor
ats907InhibitorexperimentalSmall moleculeROCK2 inhibitor
belumosudil (Rezurock)InhibitorapprovedSmall moleculeRho-associated protein kinase 2 inhibitor
cethrinInhibitorexperimentalSmall moleculeROCK2 inhibitor
fasudilInhibitorexperimentalSmall moleculeROCK2 inhibitor
gns-3545InhibitorexperimentalSmall moleculeROCK2 inhibitor
gv101InhibitorexperimentalSmall moleculeROCK2 inhibitor
opl-0401InhibitorexperimentalSmall moleculeROCK2 inhibitor
ripasudil (Glanatec)InhibitorexperimentalSmall moleculeROCK2 inhibitor
roc-101InhibitorexperimentalSmall moleculeROCK2 inhibitor
tdi01InhibitorexperimentalSmall moleculeROCK2 inhibitor
tq05105InhibitorexperimentalSmall moleculeROCK2 inhibitor
ZelasudilInhibitorexperimentalSmall moleculeROCK2 inhibitor