← Mechanisms of action
Somatostatin receptor
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (19)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| octreotide (sandostatin) | Agonist | approved | Peptide | Somatostatin receptor agonist |
| somatostatin | Agonist | experimental | Recombinant protein | Somatostatin receptor agonist |
| octreotate | Antagonist | experimental | Small molecule | Somatostatin receptor antagonist |
| [18f]-fet-βag-toca | Binding agent | experimental | Small molecule | Somatostatin receptor binding agent |
| [68ga]ga-dota-cys-ath001 | Binding agent | experimental | Small molecule | Somatostatin receptor binding agent |
| ga-68-dota-toc (Ga-68-dota-toc) | Binding agent | approved | Small molecule | Somatostatin receptor binding agent |
| lutetium dotatate lu-177 (Lutathera) | Binding agent | approved | Small molecule | Somatostatin receptor binding agent |
| satoreotide tetraxetan | Binding agent | experimental | Peptide | Somatostatin receptor binding agent |
| 90y-smt487 | Radiodepletion | experimental | Peptide | Somatostatin receptor radiodepletion |
| [68ga]ga-dota-h2d3 | Radiopharmaceutical | experimental | Small molecule | Somatostatin receptor radiopharmaceutical |
| [68ga]ga-nota-g5 | Radiopharmaceutical | experimental | Small molecule | Somatostatin receptor radiopharmaceutical |
| 18f-alf-nota-octreotide | Radiopharmaceutical | experimental | Peptide | Somatostatin receptor radiopharmaceutical |
| 68ga-g21 | Radiopharmaceutical | experimental | Peptide | Somatostatin receptor radiopharmaceutical |
| 68ga-r10602 | Radiopharmaceutical | experimental | Small molecule | Somatostatin receptor radiopharmaceutical |
| cu-64 sartate | Radiopharmaceutical | experimental | Small molecule | Somatostatin receptor radiopharmaceutical |
| cu-67 sartate | Radiopharmaceutical | experimental | Small molecule | Somatostatin receptor radiopharmaceutical |
| ga 68-edotreotide | Radiopharmaceutical | experimental | Small molecule | Somatostatin receptor radiopharmaceutical |
| lu-177-dota-octreotide | Radiopharmaceutical | experimental | Peptide | Somatostatin receptor radiopharmaceutical |
| satoreotide trizoxetan | Radiopharmaceutical | experimental | Peptide | Somatostatin receptor radiopharmaceutical |