← Mechanisms of action

Somatostatin receptor

PROTEIN FAMILYHomo sapiens

Linked proteins

Drugs acting on this target (19)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
octreotide (sandostatin)AgonistapprovedPeptideSomatostatin receptor agonist
somatostatinAgonistexperimentalRecombinant proteinSomatostatin receptor agonist
octreotateAntagonistexperimentalSmall moleculeSomatostatin receptor antagonist
[18f]-fet-βag-tocaBinding agentexperimentalSmall moleculeSomatostatin receptor binding agent
[68ga]ga-dota-cys-ath001Binding agentexperimentalSmall moleculeSomatostatin receptor binding agent
ga-68-dota-toc (Ga-68-dota-toc)Binding agentapprovedSmall moleculeSomatostatin receptor binding agent
lutetium dotatate lu-177 (Lutathera)Binding agentapprovedSmall moleculeSomatostatin receptor binding agent
satoreotide tetraxetanBinding agentexperimentalPeptideSomatostatin receptor binding agent
90y-smt487RadiodepletionexperimentalPeptideSomatostatin receptor radiodepletion
[68ga]ga-dota-h2d3RadiopharmaceuticalexperimentalSmall moleculeSomatostatin receptor radiopharmaceutical
[68ga]ga-nota-g5RadiopharmaceuticalexperimentalSmall moleculeSomatostatin receptor radiopharmaceutical
18f-alf-nota-octreotideRadiopharmaceuticalexperimentalPeptideSomatostatin receptor radiopharmaceutical
68ga-g21RadiopharmaceuticalexperimentalPeptideSomatostatin receptor radiopharmaceutical
68ga-r10602RadiopharmaceuticalexperimentalSmall moleculeSomatostatin receptor radiopharmaceutical
cu-64 sartateRadiopharmaceuticalexperimentalSmall moleculeSomatostatin receptor radiopharmaceutical
cu-67 sartateRadiopharmaceuticalexperimentalSmall moleculeSomatostatin receptor radiopharmaceutical
ga 68-edotreotideRadiopharmaceuticalexperimentalSmall moleculeSomatostatin receptor radiopharmaceutical
lu-177-dota-octreotideRadiopharmaceuticalexperimentalPeptideSomatostatin receptor radiopharmaceutical
satoreotide trizoxetanRadiopharmaceuticalexperimentalPeptideSomatostatin receptor radiopharmaceutical