← Mechanisms of action

SSTR2

SINGLE PROTEINHomo sapiens
Preferred name: Somatostatin receptor 2 ChEMBL ↗

Linked proteins

Drugs acting on this target (16)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
225ac-sso110AgonistexperimentalPeptideSSTR2 agonist
lanreotide (somatuline depot)AgonistapprovedPeptideSSTR2 agonist
PaltusotineAgonistapprovedSmall moleculeSomatostatin receptor 2 agonist
pasireotide (signifor)AgonistapprovedPeptideSSTR2 agonist
vapreotidumAgonistexperimentalPeptideSSTR2 agonist
veldoreotideAgonistexperimentalPeptideSomatostatin receptor 2 agonist
al18f-nota-lm3AntagonistexperimentalSmall moleculeSSTR2 antagonist
zt-01AntagonistexperimentalSmall moleculeSSTR2 antagonist
in-111 dotatateBinding agentexperimentalPeptideSSTR2 binding agent
mb0151InhibitorexperimentalSmall moleculeSSTR2 inhibitor
pen-221InhibitorexperimentalmAbSSTR2 inhibitor
xmab18087InhibitorexperimentalmAbSSTR2 inhibitor
y90 edotreotideInhibitorexperimentalmAbSSTR2 inhibitor
ryz401RadiodepletionexperimentalSmall moleculeSSTR2 radiodepletion
68ga-fl-031RadiopharmaceuticalexperimentalPeptideSSTR2 radiopharmaceutical
68ga-tate-rgdRadiopharmaceuticalexperimentalPeptideSSTR2 radiopharmaceutical