← Mechanisms of action

Hepatitis C virus serine protease, NS3/NS4A

PROTEIN COMPLEXHepatitis C virus

Linked proteins

Drugs acting on this target (21)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
danoprevirAntagonistexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A antagonist
glecaprevir (Mavyret)AntagonistapprovedSmall moleculeHepatitis C virus serine protease, NS3/NS4A antagonist
paritaprevir (viekira pak)AntagonistapprovedSmall moleculeHepatitis C virus serine protease, NS3/NS4A antagonist
asunaprevirInhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
boceprevir (victrelis)InhibitorapprovedSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
bzf961InhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
ciluprevirInhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
danoprevirInhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
faldaprevirInhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
furaprevirInhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
glecaprevir (Mavyret)InhibitorapprovedSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
grazoprevir (zepatier)InhibitorapprovedSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
gs-9256InhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
narlaprevirInhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
paritaprevir (viekira pak)InhibitorapprovedSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
simeprevir (olysio)InhibitorapprovedSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
sovaprevirInhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
telaprevir (incivek)InhibitorapprovedSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
vaniprevirInhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
vedroprevirInhibitorexperimentalSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor
voxilaprevir (Vosevi)InhibitorapprovedSmall moleculeHepatitis C virus serine protease, NS3/NS4A inhibitor