← Mechanisms of action
Glutamate NMDA receptor; GRIN1/GRIN2A
PROTEIN COMPLEXHomo sapiens
Linked proteins
Drugs acting on this target (5)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| cyclopropane | Antagonist | marketed | Small molecule | Glutamate NMDA receptor; GRIN1/GRIN2A antagonist |
| ketobemidone (Ketogan) | Antagonist | experimental | Small molecule | Glutamate NMDA receptor; GRIN1/GRIN2A antagonist |
| bupivacaine (Exparel) | Inhibitor | experimental | Small molecule | Glutamate NMDA receptor; GRIN1/GRIN2A inhibitor |
| ifenprodil | Inhibitor | experimental | Small molecule | Glutamate NMDA receptor; GRIN1/GRIN2A inhibitor |
| sage-718 | Inhibitor | experimental | Small molecule | Glutamate NMDA receptor; GRIN1/GRIN2A inhibitor |