← Mechanisms of action
Integrin alpha-V/beta-3
PROTEIN COMPLEXHomo sapiens
Linked proteins
Drugs acting on this target (6)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| atn-161 | Antagonist | experimental | Peptide | Integrin alpha-V/beta-3 antagonist |
| cilengitide | Antagonist | experimental | Peptide | Integrin alpha-V/beta-3 antagonist |
| etaracizumab (abegrin) | Antagonist | experimental | mAb | Integrin alpha-V/beta-3 antagonist |
| intetumumab | Antagonist | experimental | mAb | Integrin alpha-V/beta-3 antagonist |
| abciximab (Reopro) | Inhibitor | approved | mAb | Integrin alpha-V/beta-3 inhibitor |
| abituzumab | Inhibitor | experimental | mAb | Integrin alpha-V/beta-3 inhibitor |