← Mechanisms of action
BRD2
SINGLE PROTEINHomo sapiens
Preferred name: Bromodomain-containing protein 2 ChEMBL ↗
Linked proteins
Drugs acting on this target (17)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| abbv-744 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| birabresib | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| br3409 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| cc-95775 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| ep31670 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| ft-1101 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| gsk2820151 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| gsk3358699 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| jab-8263 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| mivebresib | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| molibresib | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| odm-207 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| plx51107 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| tqb3617 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| Trotabresib | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| vyn201 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |
| zen003694 | Inhibitor | experimental | Small molecule | BRD2 inhibitor |