← Mechanisms of action
Bromodomain and extra-terminal motif (BET)
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (5)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| apabetalone | Inhibitor | experimental | Small molecule | Bromodomain and extra-terminal motif (BET) inhibitor |
| birabresib | Inhibitor | experimental | Small molecule | Bromodomain and extra-terminal motif (BET) inhibitor |
| fostemsavir (Rukobia) | Inhibitor | approved | Small molecule | Bromodomain and extra-terminal motif (BET) inhibitor |
| molibresib | Inhibitor | experimental | Small molecule | Bromodomain and extra-terminal motif (BET) inhibitor |
| ro6870810 | Inhibitor | experimental | Small molecule | Bromodomain and extra-terminal motif (BET) inhibitor |