← Mechanisms of action
F2R
SINGLE PROTEINHomo sapiens
Preferred name: Proteinase-activated receptor 1 ChEMBL ↗
Linked proteins
Drugs acting on this target (4)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| atopaxar | Antagonist | experimental | Small molecule | F2R antagonist |
| vorapaxar (zontivity) | Antagonist | approved | Small molecule | F2R antagonist |
| pz-128 | Inhibitor | experimental | Small molecule | Proteinase-activated receptor 1 inhibitor |
| rigosertib | Inhibitor | experimental | Small molecule | F2R inhibitor |