← Mechanisms of action

VDR

SINGLE PROTEINHomo sapiens
Preferred name: Vitamin D receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (24)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
2-methylene-19-nor-(20s)-1,25-dihydroxyvitamin d3AgonistexperimentalSmall moleculeVDR agonist
24,25-dihydroxycholecalciferolAgonistexperimentalSmall moleculeVDR agonist
alfacalcidolAgonistexperimentalSmall moleculeVDR agonist
becocalcidiolAgonistexperimentalSmall moleculeVDR agonist
calcifediolAgonistapprovedSmall moleculeVDR agonist
calcipotriene (dovonex)AgonistapprovedSmall moleculeVDR agonist
calcipotriolAgonistexperimentalSmall moleculeVDR agonist
calcitriol (rocaltrol)AgonistapprovedSmall moleculeVDR agonist
card-024AgonistexperimentalSmall moleculeVDR agonist
cta018AgonistexperimentalSmall moleculeVDR agonist
dihydrotachysterolAgonistexperimentalSmall moleculeVDR agonist
doxercalciferol (hectorol)AgonistapprovedSmall moleculeVDR agonist
eldecalcitolAgonistexperimentalSmall moleculeVDR agonist
elocalcitolAgonistexperimentalSmall moleculeVDR agonist
ergocalciferol (drisdol)AgonistapprovedSmall moleculeVDR agonist
inecalcitolAgonistexperimentalSmall moleculeVDR agonist
leo80122AgonistexperimentalSmall moleculeVDR agonist
paricalcitol (zemplar)AgonistapprovedSmall moleculeVDR agonist
pefcalcitolAgonistexperimentalSmall moleculeVDR agonist
ro-23-7553AgonistexperimentalSmall moleculeVDR agonist
seocalcitolAgonistexperimentalSmall moleculeVDR agonist
tacalcitolAgonistexperimentalSmall moleculeVDR agonist
vitamin d3InhibitorapprovedSmall moleculeVDR inhibitor
vs-105ModulatorexperimentalSmall moleculeVDR modulator