← Mechanisms of action
VDR
SINGLE PROTEINHomo sapiens
Preferred name: Vitamin D receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (24)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| 2-methylene-19-nor-(20s)-1,25-dihydroxyvitamin d3 | Agonist | experimental | Small molecule | VDR agonist |
| 24,25-dihydroxycholecalciferol | Agonist | experimental | Small molecule | VDR agonist |
| alfacalcidol | Agonist | experimental | Small molecule | VDR agonist |
| becocalcidiol | Agonist | experimental | Small molecule | VDR agonist |
| calcifediol | Agonist | approved | Small molecule | VDR agonist |
| calcipotriene (dovonex) | Agonist | approved | Small molecule | VDR agonist |
| calcipotriol | Agonist | experimental | Small molecule | VDR agonist |
| calcitriol (rocaltrol) | Agonist | approved | Small molecule | VDR agonist |
| card-024 | Agonist | experimental | Small molecule | VDR agonist |
| cta018 | Agonist | experimental | Small molecule | VDR agonist |
| dihydrotachysterol | Agonist | experimental | Small molecule | VDR agonist |
| doxercalciferol (hectorol) | Agonist | approved | Small molecule | VDR agonist |
| eldecalcitol | Agonist | experimental | Small molecule | VDR agonist |
| elocalcitol | Agonist | experimental | Small molecule | VDR agonist |
| ergocalciferol (drisdol) | Agonist | approved | Small molecule | VDR agonist |
| inecalcitol | Agonist | experimental | Small molecule | VDR agonist |
| leo80122 | Agonist | experimental | Small molecule | VDR agonist |
| paricalcitol (zemplar) | Agonist | approved | Small molecule | VDR agonist |
| pefcalcitol | Agonist | experimental | Small molecule | VDR agonist |
| ro-23-7553 | Agonist | experimental | Small molecule | VDR agonist |
| seocalcitol | Agonist | experimental | Small molecule | VDR agonist |
| tacalcitol | Agonist | experimental | Small molecule | VDR agonist |
| vitamin d3 | Inhibitor | approved | Small molecule | VDR inhibitor |
| vs-105 | Modulator | experimental | Small molecule | VDR modulator |