← Mechanisms of action
TLR7
SINGLE PROTEINHomo sapiens
Preferred name: Toll-like receptor 7 ChEMBL ↗
Linked proteins
Drugs acting on this target (44)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| lfx453 | Activator | experimental | Small molecule | TLR7 activator |
| vesatolimod | Activator | experimental | Small molecule | Toll-like receptor 7 activator |
| 1v270 | Agonist | experimental | Small molecule | TLR7 agonist |
| 3m-05-af | Agonist | experimental | Vaccine | TLR7 agonist |
| 3m-052-af | Agonist | experimental | Small molecule | TLR7 agonist |
| al-034 | Agonist | experimental | Small molecule | TLR7 agonist |
| ana773 | Agonist | experimental | Small molecule | TLR7 agonist |
| apr002 | Agonist | experimental | Small molecule | TLR7 |
| apr003 | Agonist | experimental | Small molecule | TLR7 agonist |
| azd8848 | Agonist | experimental | Small molecule | TLR7 agonist |
| bdb001 | Agonist | experimental | Small molecule | TLR7 agonist |
| bdb018 | Agonist | experimental | Small molecule | TLR7 agonist |
| bm201 | Agonist | experimental | Small molecule | TLR7 agonist |
| bnt411 | Agonist | experimental | Small molecule | TLR7 agonist |
| can1012 | Agonist | experimental | Small molecule | TLR7 agonist |
| cpg-52852 | Agonist | experimental | Small molecule | Toll-like receptor 7 agonist |
| dsp-0509 | Agonist | experimental | Small molecule | TLR7 agonist |
| dsp-0546lp | Agonist | experimental | Small molecule | TLR7 agonist |
| eik1001 | Agonist | experimental | Small molecule | TLR7 agonist |
| gsk2445053 | Agonist | experimental | Small molecule | TLR7 agonist |
| imiquimod (aldara) | Agonist | approved | Small molecule | TLR7 agonist |
| ini-4001 | Agonist | experimental | Small molecule | TLR7 agonist |
| lhc165 | Agonist | experimental | Small molecule | TLR7 agonist |
| medi9197 | Agonist | experimental | Small molecule | TLR7 agonist |
| nktr-262 | Agonist | experimental | Small molecule | TLR7 agonist |
| pf-04878691 | Agonist | experimental | Small molecule | TLR7 agonist |
| pf-08046037 | Agonist | experimental | mAb | TLR7 agonist |
| resiquimod | Agonist | experimental | Small molecule | Toll-like receptor 7 agonist |
| ro6864018 | Agonist | experimental | Small molecule | TLR7 agonist |
| ro6870868 | Agonist | experimental | Small molecule | TLR7 agonist |
| ro7020531 | Agonist | experimental | Small molecule | TLR7 agonist |
| ro7119929 | Agonist | experimental | Small molecule | TLR7 agonist |
| shr2150 | Agonist | experimental | Small molecule | TLR7 agonist |
| tq-a3334 | Agonist | experimental | Small molecule | TLR7 agonist |
| tqa3334 | Agonist | experimental | Small molecule | TLR7 agonist |
| transcon tlr7/8 agonist | Agonist | experimental | Recombinant protein | TLR7 agonist |
| vesatolimod | Agonist | experimental | Small molecule | TLR7 agonist |
| cpg 52364 | Antagonist | experimental | Small molecule | TLR7 antagonist |
| ds-7011a | Antagonist | experimental | Small molecule | TLR7 antagonist |
| e6742 | Antagonist | experimental | Small molecule | TLR7 antagonist |
| enpatoran | Antagonist | experimental | Small molecule | Toll-like receptor 7 antagonist |
| hydroxychloroquine (plaquenil) | Antagonist | approved | Small molecule | TLR7 antagonist |
| afimetoran | Inhibitor | experimental | Small molecule | TLR7 inhibitor |
| mhv370 | Inhibitor | experimental | Small molecule | TLR7 inhibitor |