← Mechanisms of action
TLR9
SINGLE PROTEINHomo sapiens
Preferred name: Toll-like receptor 9 ChEMBL ↗
Linked proteins
Drugs acting on this target (29)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| cobitolimod | Activator | experimental | Nucleic acid | TLR9 activator |
| mis416 | Activator | experimental | Small molecule | TLR9 activator |
| agatolimod | Agonist | experimental | Small molecule | TLR9 agonist |
| bl-7040 | Agonist | experimental | Nucleic acid | TLR9 agonist |
| Cavrotolimod | Agonist | experimental | Small molecule | TLR9 agonist |
| cobitolimod | Agonist | experimental | Nucleic acid | Toll-like receptor 9 agonist |
| cpg 10104 | Agonist | experimental | Biological | TLR9 agonist |
| cpg 7909 | Agonist | experimental | Small molecule | TLR9 agonist |
| cpg 7909 oligodeoxynucleotide | Agonist | experimental | Vaccine | TLR9 agonist |
| cpg-odn | Agonist | experimental | Nucleic acid | TLR9 |
| cpg-oligonucleotide | Agonist | experimental | Nucleic acid | TLR9 agonist |
| cpg10101 | Agonist | experimental | Biological | TLR9 agonist |
| cyt003-qbg10 | Agonist | experimental | Small molecule | TLR9 agonist |
| emd 1201081 | Agonist | experimental | Nucleic acid | TLR9 agonist |
| gnkg168 | Agonist | experimental | Peptide | TLR9 agonist |
| imo-2125 | Agonist | experimental | Small molecule | TLR9 agonist |
| lefitolimod | Agonist | experimental | Nucleic acid | Toll-like receptor 9 agonist |
| pul-042 | Agonist | experimental | Small molecule | TLR9 agonist |
| sd-101 | Agonist | experimental | Small molecule | TLR9 agonist |
| tilsotolimod | Agonist | experimental | mAb | Toll-like receptor 9 agonist |
| cpg 52364 | Antagonist | experimental | Small molecule | TLR9 antagonist |
| hydroxychloroquine (plaquenil) | Antagonist | approved | Small molecule | TLR9 antagonist |
| imo-8400 | Antagonist | experimental | Small molecule | TLR9 antagonist |
| cpg-stat3 sirna cas3/ss3 | Antisense inhibitor | experimental | Nucleic acid | TLR9 antisense inhibitor |
| azd1419 | Inhibitor | experimental | Nucleic acid | TLR9 inhibitor |
| bl-1021 | Inhibitor | experimental | Small molecule | TLR9 inhibitor |
| cmp-001 | Inhibitor | experimental | mAb | TLR9 inhibitor |
| cpg 1018 | Inhibitor | experimental | mAb | TLR9 inhibitor |
| tilsotolimod | Inhibitor | experimental | mAb | TLR9 inhibitor |