← Mechanisms of action

TLR9

SINGLE PROTEINHomo sapiens
Preferred name: Toll-like receptor 9 ChEMBL ↗

Linked proteins

Drugs acting on this target (29)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
cobitolimodActivatorexperimentalNucleic acidTLR9 activator
mis416ActivatorexperimentalSmall moleculeTLR9 activator
agatolimodAgonistexperimentalSmall moleculeTLR9 agonist
bl-7040AgonistexperimentalNucleic acidTLR9 agonist
CavrotolimodAgonistexperimentalSmall moleculeTLR9 agonist
cobitolimodAgonistexperimentalNucleic acidToll-like receptor 9 agonist
cpg 10104AgonistexperimentalBiologicalTLR9 agonist
cpg 7909AgonistexperimentalSmall moleculeTLR9 agonist
cpg 7909 oligodeoxynucleotideAgonistexperimentalVaccineTLR9 agonist
cpg-odnAgonistexperimentalNucleic acidTLR9
cpg-oligonucleotideAgonistexperimentalNucleic acidTLR9 agonist
cpg10101AgonistexperimentalBiologicalTLR9 agonist
cyt003-qbg10AgonistexperimentalSmall moleculeTLR9 agonist
emd 1201081AgonistexperimentalNucleic acidTLR9 agonist
gnkg168AgonistexperimentalPeptideTLR9 agonist
imo-2125AgonistexperimentalSmall moleculeTLR9 agonist
lefitolimodAgonistexperimentalNucleic acidToll-like receptor 9 agonist
pul-042AgonistexperimentalSmall moleculeTLR9 agonist
sd-101AgonistexperimentalSmall moleculeTLR9 agonist
tilsotolimodAgonistexperimentalmAbToll-like receptor 9 agonist
cpg 52364AntagonistexperimentalSmall moleculeTLR9 antagonist
hydroxychloroquine (plaquenil)AntagonistapprovedSmall moleculeTLR9 antagonist
imo-8400AntagonistexperimentalSmall moleculeTLR9 antagonist
cpg-stat3 sirna cas3/ss3Antisense inhibitorexperimentalNucleic acidTLR9 antisense inhibitor
azd1419InhibitorexperimentalNucleic acidTLR9 inhibitor
bl-1021InhibitorexperimentalSmall moleculeTLR9 inhibitor
cmp-001InhibitorexperimentalmAbTLR9 inhibitor
cpg 1018InhibitorexperimentalmAbTLR9 inhibitor
tilsotolimodInhibitorexperimentalmAbTLR9 inhibitor