← Mechanisms of action

GCG

SINGLE PROTEINHomo sapiens
Preferred name: Glucagon ChEMBL ↗

Linked proteins

Drugs acting on this target (12)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
mod-6031ActivatorexperimentalPeptideGCG activator
oxyntomodulinActivatorexperimentalRecombinant proteinGCG activator
bi 1820237AgonistexperimentalRecombinant proteinGCG agonist
cotadutideAgonistexperimentalPeptideGCG agonist
dasiglucagon (Zegalogue)AgonistapprovedSmall moleculeGCG agonist
efpeglenatideAgonistexperimentalPeptideGCG agonist
mazdutideAgonistexperimentalPeptideGCG agonist
oap-189AgonistexperimentalPeptideGCG agonist
sar438544AgonistexperimentalSmall moleculeGCG agonist
sar441255AgonistexperimentalPeptideGCG agonist
ecc5004AntagonistexperimentalSmall moleculeGLP-1
exendin (9-39)AntagonistexperimentalPeptideGCG antagonist