← Mechanisms of action
GCG
SINGLE PROTEINHomo sapiens
Preferred name: Glucagon ChEMBL ↗
Linked proteins
Drugs acting on this target (12)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| mod-6031 | Activator | experimental | Peptide | GCG activator |
| oxyntomodulin | Activator | experimental | Recombinant protein | GCG activator |
| bi 1820237 | Agonist | experimental | Recombinant protein | GCG agonist |
| cotadutide | Agonist | experimental | Peptide | GCG agonist |
| dasiglucagon (Zegalogue) | Agonist | approved | Small molecule | GCG agonist |
| efpeglenatide | Agonist | experimental | Peptide | GCG agonist |
| mazdutide | Agonist | experimental | Peptide | GCG agonist |
| oap-189 | Agonist | experimental | Peptide | GCG agonist |
| sar438544 | Agonist | experimental | Small molecule | GCG agonist |
| sar441255 | Agonist | experimental | Peptide | GCG agonist |
| ecc5004 | Antagonist | experimental | Small molecule | GLP-1 |
| exendin (9-39) | Antagonist | experimental | Peptide | GCG antagonist |