← Mechanisms of action
ERG11
SINGLE PROTEINCandida albicans (strain SC5314 / ATCC MYA-2876) (Yeast)
Preferred name: Cytochrome P450 51 ChEMBL ↗
Linked proteins
Drugs acting on this target (17)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| butoconazole (Femstat) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| econazole (spectazole) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| fluconazole (diflucan) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| fosravuconazole | Inhibitor | experimental | Small molecule | ERG11 inhibitor |
| itraconazole (sporanox) | Inhibitor | approved | Small molecule | Cytochrome P450 51 inhibitor |
| ketoconazole (nizoral) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| luliconazole (luzu) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| miconazole (monistat) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| oxiconazole (oxistat) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| posaconazole (noxafil) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| ravuconazole | Inhibitor | experimental | Small molecule | ERG11 inhibitor |
| sertaconazole (ertaczo) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| sulconazole (exelderm) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| terconazole (terazol) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| tioconazole (tz-3) | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| urea | Inhibitor | approved | Small molecule | ERG11 inhibitor |
| voriconazole (vfend) | Inhibitor | approved | Small molecule | ERG11 inhibitor |