← Mechanisms of action

CALCA

SINGLE PROTEINHomo sapiens
Preferred name: Calcitonin gene-related peptide 1 ChEMBL ↗

Linked proteins

Drugs acting on this target (11)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
IL-23/CGRP bispecific antibodyAntagonistexperimentalmAbCALCA antagonist
js010AntagonistexperimentalSmall moleculeCALCA antagonist
zavegepant (zavzpret)AntagonistapprovedSmall moleculeCALCA antagonist
amg 223InhibitorexperimentalSmall moleculeCALCA inhibitor
bi 44370InhibitorexperimentalSmall moleculeCALCA inhibitor
eptinezumab (Vyepti)InhibitorapprovedmAbCALCA
galcanezumab-gnlm (emgality)InhibitorapprovedmAbCALCA inhibitor
htl0022562InhibitorexperimentalSmall moleculeCALCA inhibitor
telcagepant potassiumInhibitorexperimentalSmall moleculeCALCA inhibitor
ub-313InhibitorexperimentalVaccineCALCA inhibitor
VazegepantInhibitorexperimentalSmall moleculeCALCA inhibitor