CDEK
← Mechanisms of action

TRPV1

SINGLE PROTEINHomo sapiens
Preferred name: Vanilloid receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (29)

Active Pharmaceutical Ingredient Mechanism Type ▲ Approval Status API Type Mechanism of Action
vanillylnonamideActivatorexperimentalSmall moleculeTRPV1 activator
ag1321001AgonistexperimentalSmall moleculeTRPV1 agonist
ResiniferatoxinAgonistexperimentalSmall moleculeTRPV1 agonist
vocacapsaicinAgonistexperimentalSmall moleculeTRPV1 agonist
zucapsaicinAgonistexperimentalSmall moleculeTRPV1 agonist
abt-102AntagonistexperimentalSmall moleculeTRPV1 antagonist
acd440AntagonistexperimentalSmall moleculeTRPV1 antagonist
amg-517AntagonistexperimentalSmall moleculeTRPV1 antagonist
azd1386AntagonistexperimentalSmall moleculeTRPV1 antagonist
bctcAntagonistexperimentalSmall moleculeTRPV1 antagonist
dwp-05195AntagonistexperimentalSmall moleculeTRPV1 antagonist
grc-6211AntagonistexperimentalSmall moleculeTRPV1 antagonist
jnj-88998377AntagonistexperimentalSmall moleculeTRPV1 antagonist
jts-653AntagonistexperimentalSmall moleculeTRPV1 antagonist
mavatrepAntagonistexperimentalSmall moleculeTRPV1 antagonist
mk-2295AntagonistexperimentalSmall moleculeTRPV1 antagonist
mr-1817AntagonistexperimentalSmall moleculeTRPV1 antagonist
pac-14028AntagonistexperimentalSmall moleculeTRPV1 antagonist
pf-3864086AntagonistexperimentalSmall moleculeTRPV1 antagonist
phe-377AntagonistexperimentalSmall moleculeTRPV1 antagonist
sb-705498AntagonistexperimentalSmall moleculeTRPV1 antagonist
syl-1001AntagonistexperimentalSmall moleculeTRPV1 antagonist
v116517AntagonistexperimentalSmall moleculeTRPV1 antagonist
xen-d0501AntagonistexperimentalSmall moleculeTRPV1 antagonist
cannabidivarinInhibitorexperimentalSmall moleculeTRPV1 inhibitor
saf-312InhibitorexperimentalSmall moleculeTRPV1 inhibitor
askc200ModulatorexperimentalSmall moleculeTRPV1 modulator
acetaminophen (tylenol)OpenerapprovedSmall moleculeTRPV1 opener
capsaicin (qutenza)OpenerapprovedSmall moleculeTRPV1 opener