← Mechanisms of action

HCRTR1

SINGLE PROTEINHomo sapiens
Preferred name: Orexin receptor 1 ChEMBL ↗

Linked proteins

Drugs acting on this target (7)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
azd4041AgonistexperimentalSmall moleculeHCRTR1 agonist
act-539313AntagonistexperimentalSmall moleculeHCRTR1 antagonist
daridorexant (Quviviq)AntagonistapprovedSmall moleculeOrexin receptor 1 antagonist
gsk649868AntagonistexperimentalSmall moleculeHCRTR1 antagonist
jnj-61393215AntagonistexperimentalSmall moleculeHCRTR1 antagonist
lemborexant (Dayvigo)AntagonistapprovedSmall moleculeHCRTR1 antagonist
cvn766InhibitorexperimentalSmall moleculeHCRTR1 inhibitor