← Mechanisms of action
Orexin receptor
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (15)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| jzp441 | Agonist | experimental | Small molecule | Orexin receptor agonist |
| tak-123 | Agonist | experimental | Small molecule | Orexin receptor agonist |
| tak-925 | Agonist | experimental | Small molecule | Orexin receptor agonist |
| tak-994 | Agonist | experimental | Small molecule | Orexin receptor agonist |
| act-462206 | Antagonist | experimental | Small molecule | Orexin receptor antagonist |
| almorexant | Antagonist | experimental | Small molecule | Orexin receptor antagonist |
| daridorexant (Quviviq) | Antagonist | approved | Small molecule | Orexin receptor antagonist |
| e2086 | Antagonist | experimental | Small molecule | Orexin receptor antagonist |
| filorexant | Antagonist | experimental | Small molecule | Orexin receptor antagonist |
| indv-2000 | Antagonist | experimental | Small molecule | Orexin receptor antagonist |
| seltorexant | Antagonist | experimental | Small molecule | Orexin receptor antagonist |
| suvorexant (belsomra) | Antagonist | approved | Small molecule | Orexin receptor antagonist |
| ts-142 | Antagonist | experimental | Small molecule | Orexin receptor antagonist |
| yzj-1139 | Antagonist | experimental | Small molecule | Orexin receptor antagonist |
| filorexant | Inhibitor | experimental | Small molecule | Orexin receptor inhibitor |