← Mechanisms of action

GCK

SINGLE PROTEINHomo sapiens
Preferred name: Hexokinase type IV ChEMBL ↗

Linked proteins

Drugs acting on this target (17)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
arry-403ActivatorexperimentalSmall moleculeGCK activator
azd1656ActivatorexperimentalSmall moleculeGCK activator
azd5658ActivatorexperimentalSmall moleculeGCK activator
azd6370ActivatorexperimentalSmall moleculeGCK activator
azd6714ActivatorexperimentalSmall moleculeGCK activator
bms-820132ActivatorexperimentalSmall moleculeGCK activator
dorzagliatinActivatorexperimentalSmall moleculeGCK activator
ds-7309ActivatorexperimentalSmall moleculeGCK activator
gk activatorActivatorexperimentalSmall moleculeGCK activator
gk1-399ActivatorexperimentalSmall moleculeGCK activator
globalagliatinActivatorexperimentalSmall moleculeGCK activator
ly-2608204ActivatorexperimentalSmall moleculeHexokinase type IV activator
mk 0941ActivatorexperimentalSmall moleculeGCK activator
pf-04991532ActivatorexperimentalSmall moleculeGCK activator
sy-004ActivatorexperimentalSmall moleculeGCK activator
tak-329ActivatorexperimentalSmall moleculeGCK activator
ttp399ActivatorexperimentalSmall moleculeGCK activator