← Mechanisms of action
SCN10A
SINGLE PROTEINHomo sapiens
Preferred name: Sodium channel protein type X alpha subunit ChEMBL ↗
Linked proteins
Drugs acting on this target (18)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| afacifenacin | Blocker | experimental | Small molecule | SCN10A blocker |
| cinchocaine (nupercaine) | Blocker | approved | Small molecule | SCN10A blocker |
| dsp-2230 | Blocker | experimental | Small molecule | SCN10A blocker |
| funapide | Blocker | experimental | Small molecule | SCN10A blocker |
| pf-04531083 | Blocker | experimental | Small molecule | SCN10A blocker |
| crobenetine | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| fz008-145 | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| hrs4800 | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| hsk55718 | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| jmkx000623 | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| khn702 | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| ltg-305 | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| ltg-321 | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| pf-06305591 | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| Relutrigine | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| suzetrigine (Journavx) | Inhibitor | approved | Small molecule | SCN10A inhibitor |
| vx-150 | Inhibitor | experimental | Small molecule | SCN10A inhibitor |
| kindolor tosylate | Modulator | experimental | Small molecule | SCN10A modulator |