← Mechanisms of action

SCN9A

SINGLE PROTEINHomo sapiens
Preferred name: Sodium channel protein type IX alpha subunit ChEMBL ↗

Linked proteins

Drugs acting on this target (16)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
olp-1002Antisense inhibitorexperimentalNucleic acidSCN9A antisense inhibitor
azd-3161BlockerexperimentalSmall moleculeSCN9A blocker
dsp-2230BlockerexperimentalSmall moleculeSCN9A blocker
funapideBlockerexperimentalSmall moleculeSCN9A blocker
pf-05089771BlockerexperimentalSmall moleculeSCN9A blocker
raxatrigineBlockerexperimentalSmall moleculeSCN9A blocker
xen-403BlockerexperimentalSmall moleculeSCN9A blocker
biib095InhibitorexperimentalSmall moleculeSCN9A inhibitor
gdc-0276InhibitorexperimentalSmall moleculeSCN9A inhibitor
gdc-0310InhibitorexperimentalSmall moleculeSCN9A inhibitor
in1011-n17InhibitorexperimentalSmall moleculeSCN9A inhibitor
pf-05186462InhibitorexperimentalSmall moleculeSCN9A inhibitor
pf-05241328InhibitorexperimentalSmall moleculeSCN9A inhibitor
st-2427InhibitorexperimentalSmall moleculeSCN9A inhibitor
kindolor tosylateModulatorexperimentalSmall moleculeSCN9A modulator
pf-05150122StabiliserexperimentalSmall moleculeSCN9A stabiliser