← Mechanisms of action
SCN9A
SINGLE PROTEINHomo sapiens
Preferred name: Sodium channel protein type IX alpha subunit ChEMBL ↗
Linked proteins
Drugs acting on this target (16)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| olp-1002 | Antisense inhibitor | experimental | Nucleic acid | SCN9A antisense inhibitor |
| azd-3161 | Blocker | experimental | Small molecule | SCN9A blocker |
| dsp-2230 | Blocker | experimental | Small molecule | SCN9A blocker |
| funapide | Blocker | experimental | Small molecule | SCN9A blocker |
| pf-05089771 | Blocker | experimental | Small molecule | SCN9A blocker |
| raxatrigine | Blocker | experimental | Small molecule | SCN9A blocker |
| xen-403 | Blocker | experimental | Small molecule | SCN9A blocker |
| biib095 | Inhibitor | experimental | Small molecule | SCN9A inhibitor |
| gdc-0276 | Inhibitor | experimental | Small molecule | SCN9A inhibitor |
| gdc-0310 | Inhibitor | experimental | Small molecule | SCN9A inhibitor |
| in1011-n17 | Inhibitor | experimental | Small molecule | SCN9A inhibitor |
| pf-05186462 | Inhibitor | experimental | Small molecule | SCN9A inhibitor |
| pf-05241328 | Inhibitor | experimental | Small molecule | SCN9A inhibitor |
| st-2427 | Inhibitor | experimental | Small molecule | SCN9A inhibitor |
| kindolor tosylate | Modulator | experimental | Small molecule | SCN9A modulator |
| pf-05150122 | Stabiliser | experimental | Small molecule | SCN9A stabiliser |