← Mechanisms of action

ADORA2A

SINGLE PROTEINHomo sapiens
Preferred name: Adenosine A2a receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (26)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
amp-579AgonistexperimentalSmall moleculeADORA2A agonist
apadenosonAgonistexperimentalSmall moleculeADORA2A agonist
BinodenosonAgonistexperimentalSmall moleculeADORA2A agonist
bvt.115959AgonistexperimentalSmall moleculeADORA2A agonist
evodenosonAgonistexperimentalSmall moleculeADORA2A agonist
gw328267xAgonistexperimentalSmall moleculeADORA2A agonist
opa-6566AgonistexperimentalSmall moleculeADORA2A agonist
regadenoson (lexiscan)AgonistapprovedSmall moleculeADORA2A agonist
sonedenosonAgonistexperimentalSmall moleculeADORA2A agonist
uk-432097AgonistexperimentalSmall moleculeADORA2A agonist
ciforadenantAntagonistexperimentalSmall moleculeAdenosine A2a receptor antagonist
ckd-512AntagonistexperimentalSmall moleculeADORA2A antagonist
ilb2109AntagonistexperimentalSmall moleculeAdenosine A2A receptor
istradefylline (Nourianz)AntagonistapprovedSmall moleculeADORA2A antagonist
pbf-509AntagonistexperimentalSmall moleculeADORA2A antagonist
pbf-999AntagonistexperimentalSmall moleculeADORA2A antagonist
preladenantAntagonistexperimentalSmall moleculeADORA2A antagonist
sch442416AntagonistexperimentalSmall moleculeADORA2A antagonist
st1535AntagonistexperimentalSmall moleculeADORA2A antagonist
tozadenantAntagonistexperimentalSmall moleculeADORA2A antagonist
v81444AntagonistexperimentalSmall moleculeADORA2A antagonist
vipadenantAntagonistexperimentalSmall moleculeADORA2A antagonist
zimberelimabAntagonistexperimentalmAbAdenosine A2a receptor antagonist
cs3005InhibitorexperimentalSmall moleculeADORA2A inhibitor
kw-6356InhibitorexperimentalSmall moleculeADORA2A inhibitor
yzj-5053InhibitorexperimentalSmall moleculeADORA2A inhibitor