← Mechanisms of action
ADORA2A
SINGLE PROTEINHomo sapiens
Preferred name: Adenosine A2a receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (26)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| amp-579 | Agonist | experimental | Small molecule | ADORA2A agonist |
| apadenoson | Agonist | experimental | Small molecule | ADORA2A agonist |
| Binodenoson | Agonist | experimental | Small molecule | ADORA2A agonist |
| bvt.115959 | Agonist | experimental | Small molecule | ADORA2A agonist |
| evodenoson | Agonist | experimental | Small molecule | ADORA2A agonist |
| gw328267x | Agonist | experimental | Small molecule | ADORA2A agonist |
| opa-6566 | Agonist | experimental | Small molecule | ADORA2A agonist |
| regadenoson (lexiscan) | Agonist | approved | Small molecule | ADORA2A agonist |
| sonedenoson | Agonist | experimental | Small molecule | ADORA2A agonist |
| uk-432097 | Agonist | experimental | Small molecule | ADORA2A agonist |
| ciforadenant | Antagonist | experimental | Small molecule | Adenosine A2a receptor antagonist |
| ckd-512 | Antagonist | experimental | Small molecule | ADORA2A antagonist |
| ilb2109 | Antagonist | experimental | Small molecule | Adenosine A2A receptor |
| istradefylline (Nourianz) | Antagonist | approved | Small molecule | ADORA2A antagonist |
| pbf-509 | Antagonist | experimental | Small molecule | ADORA2A antagonist |
| pbf-999 | Antagonist | experimental | Small molecule | ADORA2A antagonist |
| preladenant | Antagonist | experimental | Small molecule | ADORA2A antagonist |
| sch442416 | Antagonist | experimental | Small molecule | ADORA2A antagonist |
| st1535 | Antagonist | experimental | Small molecule | ADORA2A antagonist |
| tozadenant | Antagonist | experimental | Small molecule | ADORA2A antagonist |
| v81444 | Antagonist | experimental | Small molecule | ADORA2A antagonist |
| vipadenant | Antagonist | experimental | Small molecule | ADORA2A antagonist |
| zimberelimab | Antagonist | experimental | mAb | Adenosine A2a receptor antagonist |
| cs3005 | Inhibitor | experimental | Small molecule | ADORA2A inhibitor |
| kw-6356 | Inhibitor | experimental | Small molecule | ADORA2A inhibitor |
| yzj-5053 | Inhibitor | experimental | Small molecule | ADORA2A inhibitor |