← Mechanisms of action

PDGFRB

SINGLE PROTEINHomo sapiens
Preferred name: Platelet-derived growth factor receptor beta ChEMBL ↗

Linked proteins

Drugs acting on this target (24)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
aiv007InhibitorexperimentalSmall moleculePDGFRB inhibitor
anlotinibInhibitorexperimentalSmall moleculePDGFRB inhibitor
cdp-860InhibitorexperimentalmAbPDGFRB inhibitor
cep2563InhibitorexperimentalSmall moleculePDGFRB inhibitor
cgi-1842InhibitorexperimentalSmall moleculePDGFRB inhibitor
cm-082InhibitorexperimentalSmall moleculePDGFRB inhibitor
cm082InhibitorexperimentalSmall moleculePDGFRB inhibitor
d-4517.2InhibitorexperimentalSmall moleculePDGFRB inhibitor
dasatinib (sprycel)InhibitorapprovedSmall moleculePDGFRB inhibitor
imatinib (gleevec)InhibitorapprovedSmall moleculePDGFRB inhibitor
nindetanibInhibitorexperimentalSmall moleculePDGFRB inhibitor
puquitinibInhibitorexperimentalSmall moleculePDGFRB inhibitor
regn2176InhibitorexperimentalmAbPDGFRB inhibitor
rg1530InhibitorexperimentalSmall moleculePDGFRB inhibitor
sorafenib (nexavar)InhibitorapprovedSmall moleculePDGFRB inhibitor
subutinibInhibitorexperimentalSmall moleculePDGFRB inhibitor
sunitinib (sutent)InhibitorapprovedSmall moleculePlatelet-derived growth factor receptor beta inhibitor
tandutinibInhibitorexperimentalSmall moleculePDGFRB inhibitor
tcmdc-140940InhibitorexperimentalSmall moleculePDGFRB inhibitor
telatinibInhibitorexperimentalSmall moleculePDGFRB inhibitor
telatinib mesylateInhibitorexperimentalSmall moleculePDGFRB inhibitor
tg-100801InhibitorexperimentalSmall moleculePDGFRB inhibitor
tivozanib (Fotivda)InhibitorapprovedSmall moleculePlatelet-derived growth factor receptor beta inhibitor
zsp1603InhibitorexperimentalSmall moleculePDGFRB inhibitor