← Mechanisms of action

GRIN3A

SINGLE PROTEINHomo sapiens
Preferred name: Glutamate [NMDA] receptor subunit 3A ChEMBL ↗

Linked proteins

Drugs acting on this target (20)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
ctp-692AgonistexperimentalSmall moleculeGRIN3A agonist
ewo1AgonistexperimentalSmall moleculeGRIN3A agonist
nyx-2925AgonistexperimentalSmall moleculeGRIN3A agonist
np10679Allosteric antagonistexperimentalSmall moleculeGRIN3A allosteric antagonist
azd6423AntagonistexperimentalSmall moleculeGRIN3A antagonist
bms-866949AntagonistexperimentalSmall moleculeGRIN3A antagonist
Flupirtine (katadolon)AntagonistexperimentalSmall moleculeGRIN3A antagonist
NelonemdazAntagonistexperimentalSmall moleculeGRIN3A antagonist
neramexaneAntagonistexperimentalSmall moleculeGRIN3A antagonist
perzinfotelAntagonistexperimentalSmall moleculeGRIN3A antagonist
fluoroethylnormemantineBinding agentexperimentalSmall moleculeGRIN3A binding agent
Caroverine (spadon)InhibitorexperimentalSmall moleculeGRIN3A inhibitor
dextromethadoneInhibitorexperimentalSmall moleculeGRIN3A inhibitor
dimiracetamInhibitorexperimentalSmall moleculeGRIN3A inhibitor
levophencynonateInhibitorexperimentalSmall moleculeGRIN3A inhibitor
opc-64005InhibitorexperimentalSmall moleculeGRIN3A inhibitor
nyx-458ModulatorexperimentalSmall moleculeGRIN3A modulator
PlazinemdorModulatorexperimentalSmall moleculeGRIN3A modulator
tllsh2910ModulatorexperimentalSmall moleculeGRIN3A modulator
ZelquistinelModulatorexperimentalSmall moleculeGRIN3A modulator