← Mechanisms of action

PPARA

SINGLE PROTEINHomo sapiens
Preferred name: Peroxisome proliferator-activated receptor alpha ChEMBL ↗

Linked proteins

Drugs acting on this target (26)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
cj-30039ActivatorexperimentalSmall moleculePPARA activator
lanifibranorActivatorexperimentalSmall moleculePPARA activator
aleglitazarAgonistexperimentalSmall moleculePPARA agonist
ave8134AgonistexperimentalSmall moleculePPARA agonist
ciprofibrateAgonistexperimentalSmall moleculePPARA agonist
clofibrate (atromid-s)AgonistapprovedSmall moleculePPARA agonist
cp-778875AgonistexperimentalSmall moleculePPARA agonist
drf-10945AgonistexperimentalSmall moleculePPARA agonist
elafibranor (IQIRVO)AgonistapprovedSmall moleculePeroxisome proliferator-activated receptor alpha agonist
fenofibrate (fenoglide)AgonistapprovedSmall moleculePPARA agonist
gemfibrozil (lopid)AgonistapprovedSmall moleculePPARA agonist
gw590735AgonistexperimentalSmall moleculePPARA agonist
imiglitazarAgonistexperimentalSmall moleculePPARA agonist
k-877AgonistexperimentalSmall moleculePPARA agonist
lobeglitazoneAgonistexperimentalSmall moleculePPARA agonist
ly-518674AgonistexperimentalSmall moleculePPARA agonist
mk-0767AgonistexperimentalSmall moleculePeroxisome proliferator-activated receptor alpha agonist
mk0767AgonistexperimentalSmall moleculePPARA agonist
muraglitazarAgonistexperimentalSmall moleculePPARA agonist
naveglitazarAgonistexperimentalSmall moleculePPARA agonist
ono-5129AgonistexperimentalSmall moleculePPARA agonist
pemafibrateAgonistexperimentalSmall moleculePeroxisome proliferator-activated receptor alpha agonist
saroglitazarAgonistexperimentalSmall moleculePeroxisome proliferator-activated receptor alpha agonist
tesaglitazarAgonistexperimentalSmall moleculePPARA agonist
zyh7AgonistexperimentalSmall moleculePPARA agonist
saroglitazarInhibitorexperimentalSmall moleculePPARA inhibitor