← Mechanisms of action
NTRK1
SINGLE PROTEINHomo sapiens
Preferred name: Nerve growth factor receptor Trk-A ChEMBL ↗
Linked proteins
Drugs acting on this target (32)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| e2511 | Activator | experimental | Small molecule | NTRK1 activator |
| cenegermin-bkbj (oxervate) | Agonist | approved | Recombinant protein | NTRK1 agonist |
| stsp-0902 | Agonist | experimental | Small molecule | NTRK1 agonist |
| vmd-928 | Allosteric antagonist | experimental | Small molecule | NTRK1 allosteric antagonist |
| bpi-28592 | Antagonist | experimental | Small molecule | NTRK1 antagonist |
| fcn-098 | Antagonist | experimental | Small molecule | NTRK1 antagonist |
| sna-120 | Antagonist | experimental | Small molecule | NTRK1 antagonist |
| tqb3558 | Antagonist | experimental | Small molecule | NTRK1 antagonist |
| vc004 | Antagonist | experimental | Small molecule | NTRK1 antagonist |
| asp7962 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| azd7451 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| ben2293 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| ct327 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| fb1003 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| fcn-011 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| gbr 900 | Inhibitor | experimental | mAb | NTRK1 inhibitor |
| gz389988 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| icp-723 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| lestaurtinib | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| milciclib | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| nov1601 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| ono-4474 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| ono-7579 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| pbi-100 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| pbi-200 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| pf-06273340 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| plx-7486 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| regorafenib (stivarga) | Inhibitor | approved | Small molecule | Nerve growth factor receptor Trk-A |
| selitrectinib | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| vm902a | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| xzp-5955 | Inhibitor | experimental | Small molecule | NTRK1 inhibitor |
| tavilermide | Partial agonist | experimental | Small molecule | NTRK1 partial agonist |