CDEK
← Mechanisms of action

GLP1R

SINGLE PROTEINHomo sapiens
Preferred name: Glucagon-like peptide 1 receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (127)

Active Pharmaceutical Ingredient Mechanism Type ▲ Approval Status API Type Mechanism of Action
blx-7006ActivatorexperimentalSmall moleculeGLP1R activator
albiglutide (tanzeum)AgonistapprovedPeptideGLP1R agonist
alv-100AgonistexperimentalPeptideGLP1R agonist
amg 786AgonistexperimentalPeptideGLP1R agonist
amycretinAgonistexperimentalRecombinant proteinGLP1R agonist
asc30AgonistexperimentalSmall moleculeGLP1R agonist
azd0186AgonistexperimentalSmall moleculeGLP1R agonist
azd9550AgonistexperimentalPeptideGLP1R agonist
beinaglutideAgonistexperimentalPeptideGLP1R agonist
bgm0504AgonistexperimentalPeptideGLP1R agonist
bionetideAgonistexperimentalPeptideGLP1R agonist
bmf-650AgonistexperimentalSmall moleculeGLP1R agonist
bms686117AgonistexperimentalPeptideGLP1R agonist
bpi-3016AgonistexperimentalPeptideGLP1R agonist
cjc-1134-pcAgonistexperimentalPeptideGLP1R agonist
cnto 3649AgonistexperimentalRecombinant proteinGLP1R agonist
cotadutideAgonistexperimentalPeptideGlucagon-like peptide 1 receptor agonist
ct-388AgonistexperimentalPeptideGLP1R agonist
ct-868AgonistexperimentalPeptideGLP1R agonist
ct-996AgonistexperimentalSmall moleculeGLP1R agonist
da-1726AgonistexperimentalPeptideGLP1R agonist
danuglipronAgonistexperimentalSmall moleculeGLP1R agonist
dapiglutideAgonistexperimentalPeptideGLP1R agonist
dd01AgonistexperimentalPeptideGLP1R agonist
dr10624AgonistexperimentalRecombinant proteinGLP1R agonist
dulaglutide (trulicity)AgonistapprovedPeptideGLP1R agonist
EcnoglutideAgonistexperimentalPeptideGLP-1R
efocipegtrutideAgonistexperimentalSmall moleculeGLP1R agonist
efpeglenatideAgonistexperimentalPeptideGLP1R agonist
exenatide (byetta)AgonistapprovedPeptideGLP1R agonist
ga-do3a-vs-cys40-exendin-4AgonistexperimentalPeptideGLP1R agonist
glp-1 9-36 amideAgonistexperimentalPeptideGLP1R agonist
glucagon-like peptide-1AgonistexperimentalPeptideGLP1R agonist
gma106AgonistexperimentalmAbGLP1R agonist
gs-4571AgonistexperimentalSmall moleculeGLP1R agonist
gsbr-1290AgonistexperimentalSmall moleculeGLP1R agonist
gx-g6AgonistexperimentalRecombinant proteinGLP1R agonist
gzr-18AgonistexperimentalPeptideGLP1R agonist
gzr102AgonistexperimentalPeptideGLP1R agonist
hdm1002AgonistexperimentalSmall moleculeGLP1R agonist
hdm1005AgonistexperimentalPeptideGLP1R agonist
hec-007AgonistexperimentalPeptideGLP1R agonist
hec88473AgonistexperimentalRecombinant proteinGLP1R agonist
hm15275AgonistexperimentalPeptideGLP1R agonist
hr17031AgonistexperimentalPeptideGLP1R agonist
hrs-4729AgonistexperimentalPeptideGLP1R agonist
hrs-7535AgonistexperimentalSmall moleculeGLP1R agonist
hrs-9531AgonistexperimentalPeptideGLP1R agonist
hrs9531AgonistexperimentalRecombinant proteinGLP1R agonist
hs-20094AgonistexperimentalPeptideGLP1R agonist
hs-20136AgonistexperimentalPeptideGLP1R agonist
hti-2088AgonistexperimentalPeptideGLP1R agonist
ibi3032AgonistexperimentalSmall moleculeGLP1R agonist
id110521156AgonistexperimentalSmall moleculeGLP1R agonist
incretinAgonistexperimentalSmall moleculeGLP1R agonist
jnj-64565111AgonistexperimentalPeptideGLP1R agonist
jy09AgonistexperimentalPeptideGLP1R agonist
kai-9531AgonistexperimentalSmall moleculeGLP1R agonist
kp405AgonistexperimentalPeptideGLP1R agonist
last 5 amino acids of glp-1AgonistexperimentalPeptideGLP1R agonist
liraglutide (victoza)AgonistapprovedPeptideGLP1R agonist
lixisenatide (adlyxin)AgonistapprovedPeptideGLP1R agonist
lotiglipronAgonistexperimentalSmall moleculeGLP1R agonist
loxenatideAgonistexperimentalPeptideGLP1R agonist
ly2428757AgonistexperimentalPeptideGLP1R agonist
ly3493269AgonistexperimentalPeptideGLP1R agonist
ly3541105AgonistexperimentalPeptideGLP1R agonist
ly6249492AgonistexperimentalSmall moleculeGLP1R agonist
maridebart cafraglutideAgonistexperimentalPeptideGLP1R agonist
mazdutideAgonistexperimentalPeptideGLP1R agonist
mbx 4291AgonistexperimentalPeptideGLP1R agonist
mdr-001AgonistexperimentalSmall moleculeGLP1R agonist
medi-4166AgonistexperimentalmAbGLP1R agonist
met097AgonistexperimentalPeptideGLP1R agonist
met233AgonistexperimentalSmall moleculeGLP1R agonist
mk-8521AgonistexperimentalPeptideGLP1R agonist
mkc253AgonistexperimentalPeptideGLP1R agonist
mwn109AgonistexperimentalPeptideGLP1R agonist
na-931AgonistexperimentalSmall moleculeGLP1R agonist
nb1001AgonistexperimentalPeptideGLP1R agonist
nn9925AgonistexperimentalSmall moleculeGLP1R agonist
nnc0113-6860AgonistexperimentalPeptideGLP1R agonist
nnc0113-6891AgonistexperimentalPeptideGLP1R agonist
nnc0650-0013AgonistexperimentalPeptideGLP1R agonist
nnc9204-1177AgonistexperimentalPeptideGLP1R agonist
nnc9204-1706 aAgonistexperimentalPeptideGLP1R agonist
NoiiglutideAgonistexperimentalPeptideGLP1R agonist
oap-189AgonistexperimentalPeptideGLP1R agonist
pb1023AgonistexperimentalRecombinant proteinGLP1R agonist
PegapamodutideAgonistexperimentalPeptideGLP1R agonist
pemvidutideAgonistexperimentalPeptideGLP1R agonist
pf-04856883AgonistexperimentalmAbGLP1R agonist
pf04603629AgonistexperimentalRecombinant proteinGLP1R agonist
ray1225AgonistexperimentalPeptideGLP1R agonist
rg7697AgonistexperimentalPeptideGLP1R agonist
rgt001-075AgonistexperimentalSmall moleculeGLP1R agonist
ro6807952AgonistexperimentalSmall moleculeGLP1R agonist
ro6811135AgonistexperimentalPeptideGLP1R agonist
rose-010AgonistexperimentalPeptideGLP1R agonist
sar441255AgonistexperimentalPeptideGLP1R agonist
semaglutide (Ozempic)AgonistapprovedPeptideGLP1R agonist
shr-1816AgonistexperimentalPeptideGLP1R agonist
supaglutideAgonistexperimentalPeptideGLP1R agonist
survodutideAgonistexperimentalPeptideGLP1R agonist
taspoglutideAgonistexperimentalPeptideGLP1R agonist
tb001AgonistexperimentalmAbGLP1R agonist
te-8105AgonistexperimentalPeptideGLP1R agonist
tern-601AgonistexperimentalSmall moleculeGLP1R agonist
tg103AgonistexperimentalRecombinant proteinGLP1R agonist
thdbh120AgonistexperimentalPeptideGLP1R agonist
tirzepatide (Mounjaro)AgonistapprovedPeptideGLP1R agonist
ttp054AgonistexperimentalSmall moleculeGLP1R agonist
ttp273AgonistexperimentalSmall moleculeGLP1R agonist
ubt251AgonistexperimentalPeptideGLP1R agonist
UtreglutideAgonistexperimentalPeptideGLP1R agonist
vct220AgonistexperimentalPeptideGLP1R agonist
vk2735AgonistexperimentalPeptideGLP1R agonist
xtl6001AgonistexperimentalPeptideGLP1R agonist
xw003AgonistexperimentalPeptideGLP1R agonist
xw014AgonistexperimentalSmall moleculeGLP1R agonist
zt003AgonistexperimentalRecombinant proteinGLP1R agonist
zyd1AgonistexperimentalPeptideGLP1R agonist
mbx 1416AntagonistexperimentalPeptideGLP1R antagonist
AvexitideAntisense inhibitorexperimentalNucleic acidGLP1R antisense inhibitor
ly3502970Partial agonistexperimentalSmall moleculeGLP1R partial agonist
111in-exendinRadiopharmaceuticalexperimentalmAbGLP1R radiopharmaceutical
68ga-nota-exendin-4RadiopharmaceuticalexperimentalPeptideGLP1R radiopharmaceutical