← Mechanisms of action
ABAT
SINGLE PROTEINHomo sapiens
Preferred name: Gamma-amino-N-butyrate transaminase ChEMBL ↗
Linked proteins
Drugs acting on this target (26)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| azd3043 | Activator | experimental | Small molecule | ABAT activator |
| enx-101 | Activator | experimental | Small molecule | ABAT activator |
| enx-102 | Activator | experimental | Small molecule | ABAT activator |
| k201 | Activator | experimental | Small molecule | ABAT activator |
| org25435 | Activator | experimental | Small molecule | ABAT activator |
| sofadil | Activator | experimental | Small molecule | ABAT activator |
| brotizolam (Lendormin) | Agonist | experimental | Small molecule | ABAT agonist |
| dextofisopam | Agonist | experimental | Small molecule | ABAT agonist |
| etifoxine (Stresam) | Agonist | experimental | Small molecule | ABAT agonist |
| Lormetazepam | Agonist | experimental | Small molecule | ABAT agonist |
| mk-0777 | Agonist | experimental | Small molecule | ABAT agonist |
| muscimol | Agonist | experimental | Small molecule | ABAT agonist |
| phenazepam | Agonist | experimental | Small molecule | ABAT agonist |
| basmisanil | Inhibitor | experimental | Small molecule | ABAT inhibitor |
| cpp-115 | Inhibitor | experimental | Small molecule | ABAT inhibitor |
| vigabatrin (sabril) | Inhibitor | approved | Small molecule | ABAT inhibitor |
| ro15-4513 | Inverse agonist | experimental | Small molecule | ABAT inverse agonist |
| Fasedienol | Modulator | experimental | Small molecule | ABAT modulator |
| gt-002 | Modulator | experimental | Small molecule | ABAT modulator |
| nora520 | Modulator | experimental | Small molecule | ABAT modulator |
| prax-114 | Modulator | experimental | Small molecule | ABAT modulator |
| zoplicone | Modulator | experimental | Small molecule | ABAT modulator |
| zuranolone (ZURZUVAE) | Modulator | approved | Small molecule | ABAT modulator |
| cvl-865 | Positive allosteric modulator | experimental | Small molecule | ABAT positive allosteric modulator |
| sage-324 | Positive allosteric modulator | experimental | Small molecule | ABAT positive allosteric modulator |
| sepranolone | Positive allosteric modulator | experimental | Small molecule | ABAT positive allosteric modulator |