← Mechanisms of action
TIGIT
SINGLE PROTEINHomo sapiens
Preferred name: T-cell immunoreceptor with Ig and ITIM domains ChEMBL ↗
Linked proteins
Drugs acting on this target (44)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ab154 | Antagonist | experimental | mAb | TIGIT antagonist |
| ab308 | Antagonist | experimental | mAb | TIGIT |
| agen1777 | Antagonist | experimental | mAb | TIGIT |
| ak127 | Antagonist | experimental | mAb | TIGIT |
| ak130 | Antagonist | experimental | mAb | TIGIT |
| asp8374 | Antagonist | experimental | mAb | TIGIT antagonist |
| AZD2936 | Antagonist | experimental | mAb | TIGIT |
| bat6005 | Antagonist | experimental | mAb | TIGIT |
| bat6021 | Antagonist | experimental | mAb | TIGIT |
| bgb-a1217 | Antagonist | experimental | mAb | TIGIT antagonist |
| bms-986442 | Antagonist | experimental | mAb | TIGIT |
| eos884448 | Antagonist | experimental | mAb | TIGIT antagonist |
| hb0036 | Antagonist | experimental | mAb | TIGIT |
| hlx301 | Antagonist | experimental | mAb | TIGIT |
| hlx53 | Antagonist | experimental | Recombinant protein | TIGIT |
| ibi321 | Antagonist | experimental | mAb | TIGIT |
| js006 | Antagonist | experimental | mAb | TIGIT |
| ly3435151 | Antagonist | experimental | mAb | TIGIT antagonist |
| omp-313m32 | Antagonist | experimental | mAb | TIGIT antagonist |
| tiraglolumab | Antagonist | experimental | mAb | TIGIT |
| tiragolumab | Antagonist | experimental | mAb | TIGIT antagonist |
| vibostolimab | Antagonist | experimental | mAb | T-cell immunoreceptor with Ig and ITIM domains antagonist |
| zg005 | Antagonist | experimental | mAb | TIGIT antagonist |
| ab154 | Inhibitor | experimental | mAb | T-cell immunoreceptor with Ig and ITIM domains inhibitor |
| bc008 | Inhibitor | experimental | mAb | TIGIT inhibitor |
| belrestotug | Inhibitor | experimental | mAb | inhibitor - TIGIT |
| belrestotug | Inhibitor | experimental | mAb | inhibitor - TIGIT |
| belrestotug | Inhibitor | experimental | mAb | inhibitor - TIGIT |
| bgb-a1217 | Inhibitor | experimental | mAb | T-cell immunoreceptor with Ig and ITIM domains inhibitor |
| bms-986207 | Inhibitor | experimental | mAb | TIGIT inhibitor |
| com902 | Inhibitor | experimental | mAb | TIGIT inhibitor |
| hb0030 | Inhibitor | experimental | mAb | inhibitor - TIGIT |
| hy07121 | Inhibitor | experimental | mAb | TIGIT inhibitor |
| ibi939 | Inhibitor | experimental | mAb | TIGIT inhibitor |
| m6223 | Inhibitor | experimental | mAb | TIGIT inhibitor |
| omp-313m32 | Inhibitor | experimental | mAb | T-cell immunoreceptor with Ig and ITIM domains inhibitor |
| pm1009 | Inhibitor | experimental | mAb | inhibitor - TIGIT |
| pm1021 | Inhibitor | experimental | mAb | inhibitor - TIGIT |
| pm1022 | Inhibitor | experimental | mAb | inhibitor - TIGIT |
| sgn-tgt | Inhibitor | experimental | mAb | TIGIT inhibitor |
| sh006 | Inhibitor | experimental | mAb | TIGIT inhibitor |
| sim0348 | Inhibitor | experimental | mAb | inhibitor - TIGIT |
| tiragolumab | Inhibitor | experimental | mAb | T-cell immunoreceptor with Ig and ITIM domains inhibitor |
| vibostolimab | Inhibitor | experimental | mAb | inhibitor - TIGIT |