← Mechanisms of action
GCGR
SINGLE PROTEINHomo sapiens
Preferred name: Glucagon receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (40)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| cotadutide | Activator | experimental | Peptide | GCGR activator |
| ga-do3a-vs-cys40-tuna-2 | Activator | experimental | Peptide | GCGR activator |
| cotadutide | Agonist | experimental | Peptide | Glucagon receptor agonist |
| dasiglucagon (Zegalogue) | Agonist | approved | Small molecule | Glucagon receptor agonist |
| dd01 | Agonist | experimental | Peptide | GCGR agonist |
| dr10624 | Agonist | experimental | Recombinant protein | GCGR agonist |
| dulaglutide (trulicity) | Agonist | approved | Peptide | Glucagon receptor agonist |
| efocipegtrutide | Agonist | experimental | Small molecule | GCGR agonist |
| glucagon | Agonist | approved | Biological | GCGR agonist |
| hec-007 | Agonist | experimental | Peptide | GCGR agonist |
| hm15136 | Agonist | experimental | Peptide | GCGR agonist |
| hm15275 | Agonist | experimental | Peptide | GCGR agonist |
| hrs-4729 | Agonist | experimental | Peptide | GCGR agonist |
| jnj-64565111 | Agonist | experimental | Peptide | GCGR agonist |
| ly3185643 | Agonist | experimental | Recombinant protein | GCGR agonist |
| mazdutide | Agonist | experimental | Peptide | GCGR agonist |
| mk-8521 | Agonist | experimental | Peptide | GCGR agonist |
| mwn109 | Agonist | experimental | Peptide | GCGR agonist |
| na-931 | Agonist | experimental | Small molecule | GCGR agonist |
| nnc0650-0013 | Agonist | experimental | Peptide | GCGR agonist |
| nnc9204-0530 | Agonist | experimental | Peptide | GCGR agonist |
| nnc9204-1177 | Agonist | experimental | Peptide | GCGR agonist |
| nnc9204-1706 a | Agonist | experimental | Peptide | GCGR agonist |
| oap-189 | Agonist | experimental | Peptide | GCGR agonist |
| pemvidutide | Agonist | experimental | Peptide | GCGR agonist |
| sar425899 | Agonist | experimental | Small molecule | GCGR agonist |
| shr-1816 | Agonist | experimental | Peptide | GCGR agonist |
| survodutide | Agonist | experimental | Peptide | GCGR agonist |
| tb001 | Agonist | experimental | mAb | GCGR agonist |
| ubt251 | Agonist | experimental | Peptide | GCGR agonist |
| xtl6001 | Agonist | experimental | Peptide | GCGR agonist |
| adomeglivant | Antagonist | experimental | Small molecule | GCGR antagonist |
| ly2393910 | Antagonist | experimental | Small molecule | GCGR antagonist |
| mk-0893 | Antagonist | experimental | Small molecule | GCGR antagonist |
| mk-3577 | Antagonist | experimental | Small molecule | Glucagon receptor antagonist |
| pf-06291874 | Antagonist | experimental | Small molecule | GCGR antagonist |
| ly3143753 | Inhibitor | experimental | Small molecule | GCGR inhibitor |
| pf-06293620 | Inhibitor | experimental | Small molecule | GCGR inhibitor |
| regn1193 | Inhibitor | experimental | mAb | GCGR inhibitor |
| remd-477 | Inhibitor | experimental | mAb | GCGR inhibitor |