← Mechanisms of action

Topoisomerase I/II

PROTEIN FAMILYHomo sapiens

Linked proteins

Drugs acting on this target (7)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
Acridine CarboxamideInhibitorexperimentalSmall moleculeTopoisomerase I/II inhibitor
amonafideInhibitorexperimentalSmall moleculeTopoisomerase I/II inhibitor
hydroxycamptothecinInhibitorexperimentalSmall moleculeTopoisomerase I/II inhibitor
iododoxorubicinInhibitorexperimentalSmall moleculeTopoisomerase I/II inhibitor
karenitecinInhibitorexperimentalSmall moleculeTopoisomerase I/II inhibitor
lapachoneInhibitorexperimentalSmall moleculeTopoisomerase I/II inhibitor
SilatecanInhibitorexperimentalSmall moleculeTopoisomerase I/II inhibitor