← Mechanisms of action
PPARG
SINGLE PROTEINHomo sapiens
Preferred name: Peroxisome proliferator-activated receptor gamma ChEMBL ↗
Linked proteins
Drugs acting on this target (45)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| Edaglitazone | Activator | experimental | Small molecule | PPARG activator |
| lanifibranor | Activator | experimental | Small molecule | PPARG activator |
| Leriglitazone | Activator | experimental | Small molecule | PPARG activator |
| puerarin | Activator | experimental | Small molecule | PPARG activator |
| aleglitazar | Agonist | experimental | Small molecule | PPARG agonist |
| ave0847 | Agonist | experimental | Small molecule | PPARG agonist |
| balsalazide (colazal) | Agonist | approved | Small molecule | PPARG agonist |
| clx-0921 | Agonist | experimental | Small molecule | PPARG agonist |
| dlbs3233 | Agonist | experimental | Botanical | PPARG agonist |
| efatutazone | Agonist | experimental | Small molecule | PPARG agonist |
| etalocib | Agonist | experimental | Small molecule | PPARG agonist |
| farglitazar | Agonist | experimental | Small molecule | PPARG agonist |
| gsk376501 | Agonist | experimental | Small molecule | PPARG agonist |
| imiglitazar | Agonist | experimental | Small molecule | PPARG agonist |
| Leriglitazone | Agonist | experimental | Small molecule | Peroxisome proliferator-activated receptor gamma agonist |
| lobeglitazone | Agonist | experimental | Small molecule | PPARG agonist |
| mk-0767 | Agonist | experimental | Small molecule | Peroxisome proliferator-activated receptor gamma agonist |
| mk0767 | Agonist | experimental | Small molecule | PPARG agonist |
| muraglitazar | Agonist | experimental | Small molecule | PPARG agonist |
| naveglitazar | Agonist | experimental | Small molecule | PPARG agonist |
| olsalazine (dipentum) | Agonist | approved | Small molecule | PPARG agonist |
| oms-405 | Agonist | experimental | Small molecule | PPARG agonist |
| ono-5129 | Agonist | experimental | Small molecule | PPARG agonist |
| pn2034 | Agonist | experimental | Small molecule | PPARG agonist |
| rivoglitazone | Agonist | experimental | Small molecule | PPARG agonist |
| rosiglitazone | Agonist | approved | Small molecule | PPARG agonist |
| saroglitazar | Agonist | experimental | Small molecule | Peroxisome proliferator-activated receptor gamma agonist |
| t3d-959 | Agonist | experimental | Small molecule | PPARG agonist |
| tesaglitazar | Agonist | experimental | Small molecule | PPARG agonist |
| troglitazone (Rezulin) | Agonist | withdrawn | Small molecule | PPARG agonist |
| bardoxolone | Antagonist | experimental | Small molecule | PPARG antagonist |
| Eucalyptol (listerine) | Inhibitor | experimental | Small molecule | PPARG inhibitor |
| fx-909 | Inhibitor | experimental | Small molecule | PPARG inhibitor |
| saroglitazar | Inhibitor | experimental | Small molecule | PPARG inhibitor |
| arhalofenate | Modulator | experimental | Small molecule | PPARG modulator |
| cb-0406 | Modulator | experimental | Small molecule | PPARG modulator |
| fk-614 | Modulator | experimental | Small molecule | PPARG modulator |
| ged-0507-34-levo | Modulator | experimental | Small molecule | PPARG modulator |
| mbx-2044 | Modulator | experimental | Small molecule | PPARG modulator |
| mk-0533 | Modulator | experimental | Small molecule | PPARG modulator |
| netoglitazone | Modulator | experimental | Small molecule | PPARG modulator |
| t131 | Modulator | experimental | Small molecule | PPARG modulator |
| balaglitazone | Partial agonist | experimental | Small molecule | PPARG partial agonist |
| dsp-8658 | Partial agonist | experimental | Small molecule | PPARG partial agonist |
| mbf-018 | Partial agonist | experimental | Small molecule | PPARG partial agonist |