← Mechanisms of action

PLG

SINGLE PROTEINHomo sapiens
Preferred name: Plasminogen ChEMBL ↗

Linked proteins

Drugs acting on this target (17)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
alteplase (Activase)ActivatorapprovedRecombinant proteinPLG activator
apsacActivatorexperimentalRecombinant proteinPLG activator
biib132ActivatorexperimentalNucleic acidPLG activator
defibrotide (defitelio)ActivatorapprovedAnimal productPLG activator
DesmoteplaseActivatorexperimentalRecombinant proteinPLG activator
dnaseActivatorexperimentalRecombinant proteinPLG activator
lt3001ActivatorexperimentalSmall moleculePLG activator
reteplase (Retavase)ActivatorapprovedRecombinant proteinPLG activator
saruplaseActivatorexperimentalRecombinant proteinPLG activator
streptokinase (streptase)ActivatorapprovedBiologicalPLG activator
tenecteplase (tnkase)ActivatorapprovedRecombinant proteinPLG activator
urokinase (kinlytic)ActivatorapprovedBiologicalPLG activator
plasminogen (Ryplazim)AgonistapprovedBiologicalPLG agonist
aminocaproic acid (amicar)InhibitorapprovedSmall moleculePLG inhibitor
aprotinin (trasylol)InhibitorwithdrawnSmall moleculePLG inhibitor
bt-114143InhibitorexperimentalSmall moleculePLG inhibitor
tranexamic acid (cyklokapron)InhibitorapprovedSmall moleculePLG inhibitor