← Mechanisms of action
Glutamate NMDA receptor
PROTEIN COMPLEX GROUPMus musculus
Linked proteins
- Glutamate receptor ionotropic, NMDA 2A (Grin2a) ↗
- Glutamate receptor ionotropic, NMDA 3B (Grin3b) ↗
- Glutamate receptor ionotropic, NMDA 2D (Grin2d) ↗
- Glutamate receptor ionotropic, NMDA 1 (Grin1) ↗
- Glutamate receptor ionotropic, NMDA 2B (Grin2b) ↗
- Glutamate receptor ionotropic, NMDA 2C (Grin2c) ↗
- Glutamate receptor ionotropic, NMDA3A (Grin3a) ↗
Drugs acting on this target (9)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| acp-211 | Antagonist | experimental | Small molecule | Glutamate NMDA receptor antagonist |
| gacyclidine | Antagonist | experimental | Small molecule | Glutamate NMDA receptor antagonist |
| kynurenic acid | Antagonist | experimental | Small molecule | Glutamate NMDA receptor antagonist |
| art5803 | Inhibitor | experimental | mAb | Glutamate NMDA receptor inhibitor |
| exv-802 | Inhibitor | experimental | Small molecule | Glutamate NMDA receptor inhibitor |
| agn-241751 | Modulator | experimental | Small molecule | Glutamate NMDA receptor modulator |
| nbi-1070770 | Negative allosteric modulator | experimental | Small molecule | Glutamate NMDA receptor negative allosteric modulator |
| sage-904 | Positive allosteric modulator | experimental | Small molecule | Glutamate NMDA receptor positive allosteric modulator |
| bnh-015b | Positive modulator | experimental | Small molecule | Glutamate NMDA receptor positive modulator |