← Mechanisms of action
MTOR
SINGLE PROTEINHomo sapiens
Preferred name: Serine/threonine-protein kinase mTOR ChEMBL ↗
Linked proteins
Drugs acting on this target (44)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| hydroxymethylbutyrate | Activator | experimental | Small molecule | MTOR activator |
| al58805 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| apitolisib | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| atg-008 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| azd-8055 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| bimiralisib | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| cc-115 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| cc-223 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| cerc-006 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| dactolisib | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| dcbci0901 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| ds-3078a | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| ds-7423 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| gdc-0349 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| gedatolisib | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| hec 68498 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| hec68498 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| kanglaite | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| ky1005 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| Lixumistat | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| ly-3023414 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| ly3023414 | Inhibitor | experimental | Small molecule | Serine/threonine-protein kinase mTOR inhibitor |
| nvp-bgt226 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| omipalisib | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| osi-027 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| palomid 529 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| panulisib | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| pentadecanoic acid | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| perhexiline maleate | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| pf-04691502 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| pf-06409577 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| pki-179 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| pqr309 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| pwt-33579 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| pwt-33587 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| ridaforolimus | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| rmc-5552 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| sapanisertib | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| sf1126 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| sirolimus (rapamune) | Inhibitor | approved | Small molecule | MTOR inhibitor |
| vistusertib | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| vs-5584 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| xl765 | Inhibitor | experimental | Small molecule | MTOR inhibitor |
| ea-230 | Stabiliser | experimental | Peptide | MTOR stabiliser |