← Mechanisms of action
CRBN
SINGLE PROTEINHomo sapiens
Preferred name: Protein cereblon ChEMBL ↗
Linked proteins
Drugs acting on this target (5)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| cft7455 | Activator | experimental | Small molecule | CRBN activator |
| cc-11006 | Inhibitor | experimental | Small molecule | CRBN inhibitor |
| Iberdomide | Inhibitor | experimental | Small molecule | CRBN inhibitor |
| Mezigdomide | Inhibitor | experimental | Small molecule | CRBN inhibitor |
| bms-986470 | Modulator | experimental | Small molecule | CRBN modulator |