picoplatin

Small moleculeexperimental

Picoplatin is a platinum-based antineoplastic agent in clinical development by Poniard Pharmaceuticals for the treatment of patients with solid tumors. — Wikipedia

Clinical trial activity

8 trials · 4 clinical orgs · 0 marketing orgs

Phase 1
5
Phase 2
5
Phase 3
1
Phase 4
0

Earliest trial started Nov 1, 2000 (NCT00016172)

Timeline

2000s

  1. Jan 1, 2000

    Earliest Phase 1 Sponsor(trial)

  2. Jan 1, 2001

    Earliest Phase 2 Sponsor(trial)

  3. Jan 1, 2007

    Earliest Phase 3 Sponsor(trial)

Indications

Mechanism of action

  • DNACROSS-LINKING AGENT

    DNA cross-linking agent

Chemistry & pharmacology

Mol. weight
376.14 g/mol
Chirality
Achiral Molecule
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • amd473
  • amd 473
  • amd-473
  • amd-473
  • amd-473
  • amminedichloro(2-methylpyridine)platinum(ii)
  • cis-amminedichloro(2-methylpyridine)platinum(ii)
  • jm473
  • jm-473
  • nx-473
  • nx-473
  • picoplatin
  • picoplatin
  • picoplatin
  • picoplatin
  • picoplatin
  • (sp-4-3)-amminedichloro(2-methylpyridine)platinium
  • (sp-4-3)-amminedichloro(2-methylpyridine)platinium
  • zd0473
  • zd 0473
  • zd-0473
  • zd-0473
  • zd-0473

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT00710697Phase 1Jun 1, 2008Poniard Pharmaceuticals
NCT00465491Phase 3Apr 1, 2007Poniard Pharmaceuticals
NCT00465725Phase 1Apr 1, 2007Poniard Pharmaceuticals
NCT00448734Phase 1/Phase 2 (Phase 2)Jun 1, 2006Poniard Pharmaceuticals
NCT00478946Phase 1/Phase 2 (Phase 2)Apr 1, 2006Poniard Pharmaceuticals
NCT00116610Phase 2Jun 1, 2005Poniard Pharmaceuticals
NCT00021008Phase 2Jul 11, 2001National Cancer Institute (NCI), University of California, Los Angeles
NCT00016172Phase 1Nov 1, 2000Cornell University, National Cancer Institute (NCI)
Showing 8 of 8 trials
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Organizations

Research & Development (4)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Poniard PharmaceuticalsFor profit6632005
National Cancer Institute (NCI)Government2022000
Cornell UniversityAcademic/Hospital1112000
University of California, Los AngelesAcademic/Hospital1112001
4 organizations
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