nop-1a

Small moleculeexperimentalImaging agent

Clinical trial activity

3 trials · 4 clinical orgs · 0 marketing orgs

Phase 1
3
Phase 2
0
Phase 3
0
Phase 4
0

Earliest trial started Sep 3, 2010 (NCT01198197)

Timeline

2010s

  1. Jan 1, 2010

    Earliest Phase 1 Sponsor(trial)

Indications

Mechanism of action

  • Unspecified targetRadiopharmaceutical

    radiopharmaceutical

Chemistry & pharmacology

Loading structure…

SMILES

CNC(=O)[C@@H](Cc1ccccc1F)CN1CCC2(CC1)OCCc1cc(F)sc12
Mol. weight
420.53 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Single Stereoisomer
Inorganic
No
Polymer
No
Imaging
11-carbon

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • nop-1a
  • nop-1a

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT03448016Early Phase 1 (Phase 1)May 27, 2016National Institute on Alcohol Abuse and Alcoholism (NIAAA), University of Pittsburgh
NCT03348384Early Phase 1 (Phase 1)Oct 30, 2014National Institute on Drug Abuse (NIDA), University of Pittsburgh
NCT01198197Early Phase 1 (Phase 1)Sep 3, 2010National Institute of Mental Health (NIMH)
Showing 3 of 3 trials
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Organizations

Research & Development (4)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
University of PittsburghAcademic/Hospital2212014
National Institute of Mental Health (NIMH)Government1112010
National Institute on Alcohol Abuse and Alcoholism (NIAAA)Government1012016
National Institute on Drug Abuse (NIDA)Government1012014
4 organizations
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