trastuzumab rezetecan
mAbexperimentalADC
Clinical trial activity
7 trials · 10 clinical orgs · 0 marketing orgs
Phase 1
0
Phase 2
7
Phase 3
0
Phase 4
0
Earliest trial started Jul 1, 2025 (NCT07047755)
Timeline
2020s
- Jan 1, 2025
Earliest Phase 2 Sponsor(trial)
Indications
Mechanism of action
ERBB2 inhibitor
Chemistry & pharmacology
- Chirality
- Single Stereoisomer
- Inorganic
- No
- Polymer
- No
- Payload
- rezetecan
Oral
No
Parenteral
No
Topical
No
Sources
- ChEMBLCHEMBL5314712 ↗
Clinical trials
| NCT ID | Phase | Start date | Sponsor(s) |
|---|---|---|---|
| NCT07309770 | Phase 2 | Dec 18, 2025 | Fudan University |
| NCT07129018 | Phase 2 | Nov 30, 2025 | Eastern Hepatobiliary Surgery Hospital, Huazhong University of Science and Technology |
| NCT07241793 | Phase 2 | Nov 20, 2025 | Guangzhou Medical University, Huazhong University of Science and Technology, Kunming Medical University, Sun Yat-Sen University |
| NCT07203729 | Phase 2 | Nov 1, 2025 | Chinese Academy of Medical Sciences |
| NCT07179939 | Phase 2 | Sep 10, 2025 | Fudan University, Hengrui Therapeutics, Inc., People's Liberation Army of China |
| NCT07100600 | Phase 2 | Aug 30, 2025 | Henan Medical University |
| NCT07047755 | Phase 2 | Jul 1, 2025 | Henan Medical University |
Showing 7 of 7 trials
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Organizations
Research & Development (10)
| Organization | Org type | Trials | As lead sponsor | Phases | Earliest year |
|---|---|---|---|---|---|
| Fudan University | Academic/Hospital | 2 | 2 | 1 | 2025 |
| Henan Medical University | Academic/Hospital | 2 | 2 | 1 | 2025 |
| Huazhong University of Science and Technology | Academic/Hospital | 2 | 1 | 1 | 2025 |
| Chinese Academy of Medical Sciences | Academic/Hospital | 1 | 1 | 1 | 2025 |
| Eastern Hepatobiliary Surgery Hospital | Academic/Hospital | 1 | 0 | 1 | 2025 |
| Guangzhou Medical University | Academic/Hospital | 1 | 0 | 1 | 2025 |
| Hengrui Therapeutics, Inc. | For profit | 1 | 0 | 1 | 2025 |
| Kunming Medical University | Academic/Hospital | 1 | 0 | 1 | 2025 |
| People's Liberation Army of China | Government | 1 | 0 | 1 | 2025 |
| Sun Yat-Sen University | Academic/Hospital | 1 | 1 | 1 | 2025 |
10 organizations
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