Pumecitinib
Small moleculeexperimental
Clinical trial activity
3 trials · 12 clinical orgs · 0 marketing orgs
Phase 1
0
Phase 2
3
Phase 3
2
Phase 4
0
Earliest trial started Mar 15, 2024 (NCT06587685)
Timeline
Indications
Mechanism of action
- Tyrosine-protein kinase JAK1INHIBITOR
JAK1 inhibitor
Chemistry & pharmacology
Loading structure…
SMILES
CC(C)S(=O)(=O)N1CC(CC#N)(n2cc(-c3ncnc4[nH]ccc34)c(N)n2)C1- Mol. weight
- 400.47 g/mol
- Lipinski Ro5
- Pass
- Rule of 3
- No
- Chirality
- Achiral Molecule
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- ChEMBLCHEMBL5314478 ↗
Clinical trials
| NCT ID | Phase | Start date | Sponsor(s) |
|---|---|---|---|
| NCT07146126 | Phase 3 | Sep 15, 2025 | Capital Medical University, Prime Gene Therapeutics Co., Ltd. |
| NCT06837233 | Phase 2 | Mar 12, 2025 | Capital Medical University, Prime Gene Therapeutics Co., Ltd. |
| NCT06587685 | Phase 3 | Mar 15, 2024 | Capital Medical University, China Medical University, Fujian Medical University, Guangzhou Medical University, Hebei University, Nanchang University, Nanyang Central Hospital, Ningbo University, Peking University, Prime Gene Therapeutics Co., Ltd., Shanxi Medical University, Southern Medical University |
Showing 3 of 3 trials
Page 1 / 1
Organizations
Research & Development (12)
| Organization | Org type | Trials | As lead sponsor | Phases | Earliest year |
|---|---|---|---|---|---|
| Capital Medical University | Academic/Hospital | 3 | 0 | 2 | 2024 |
| Prime Gene Therapeutics Co., Ltd. | For profit | 3 | 3 | 2 | 2024 |
| China Medical University | Academic/Hospital | 1 | 0 | 1 | 2024 |
| Fujian Medical University | Academic/Hospital | 1 | 0 | 1 | 2024 |
| Guangzhou Medical University | Academic/Hospital | 1 | 0 | 1 | 2024 |
| Hebei University | Academic/Hospital | 1 | 0 | 1 | 2024 |
| Nanchang University | Academic/Hospital | 1 | 0 | 1 | 2024 |
| Nanyang Central Hospital | Academic/Hospital | 1 | 0 | 1 | 2024 |
| Ningbo University | Academic/Hospital | 1 | 0 | 1 | 2024 |
| Peking University | Academic/Hospital | 1 | 0 | 1 | 2024 |
| Shanxi Medical University | Academic/Hospital | 1 | 0 | 1 | 2024 |
| Southern Medical University | Academic/Hospital | 1 | 0 | 1 | 2024 |
12 organizations
Page 1 / 1