golidocitinib
Small moleculeexperimental
Clinical trial activity
22 trials · 10 clinical orgs · 0 marketing orgs
Phase 1
10
Phase 2
21
Phase 3
1
Phase 4
0
Earliest trial started Aug 3, 2023 (NCT05963347)
Timeline
Indications
Mechanism of action
- Jak1 proteinINHIBITOR
JAK1 inhibitor
- Tyrosine-protein kinase JAK1INHIBITOR
Tyrosine-protein kinase JAK1 inhibitor
Chemistry & pharmacology
Loading structure…
SMILES
COc1nn(C)cc1Nc1nccc(-c2c[nH]c3c(NC(=O)[C@@H](C)N4CCN(C)CC4)cccc23)n1- Mol. weight
- 489.58 g/mol
- Lipinski Ro5
- Pass
- Rule of 3
- No
- Chirality
- Single Stereoisomer
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- ChEMBLCHEMBL4577523 ↗
Clinical trials
| NCT ID | Phase | Start date | Sponsor(s) |
|---|---|---|---|
| NCT07303881 | Phase 2 | Feb 28, 2026 | Guangzhou Medical University |
| NCT07279584 | Phase 2 | Dec 20, 2025 | Jiao Tong University |
| NCT07297550 | Phase 1/Phase 2 (Phase 2) | Dec 15, 2025 | China Academy of Chinese Medical Sciences |
| NCT07209163 | Phase 1/Phase 2 (Phase 2) | Oct 31, 2025 | Jiao Tong University |
| NCT07196163 | Phase 1/Phase 2 (Phase 2) | Oct 30, 2025 | Peking University |
| NCT07110103 | Phase 2 | Aug 15, 2025 | Chinese Academy of Medical Sciences, Dizal (Jiangsu) Pharmaceutical Co., Ltd. |
| NCT07093710 | Phase 1/Phase 2 (Phase 2) | Aug 1, 2025 | Sun Yat-Sen University |
| NCT07032532 | Phase 2 | Jul 31, 2025 | Sun Yat-Sen University |
| NCT07081607 | Phase 2 | Jul 15, 2025 | Jiao Tong University |
| NCT06966154 | Phase 1/Phase 2 (Phase 2) | May 26, 2025 | Fudan University |
| NCT06969612 | Phase 1 | May 15, 2025 | Peking University |
| NCT06630091 | Phase 2 | Mar 28, 2025 | University of Texas at Houston |
| NCT06855823 | Phase 1/Phase 2 (Phase 2) | Jan 14, 2025 | Sun Yat-Sen University |
| NCT06733051 | Phase 2 | Dec 31, 2024 | Sun Yat-Sen University |
| NCT06757387 | Phase 1/Phase 2 (Phase 2) | Dec 30, 2024 | Peking University |
| NCT06690671 | Phase 1/Phase 2 (Phase 2) | Dec 15, 2024 | Jiao Tong University |
| NCT06701344 | Phase 2 | Dec 4, 2024 | Jiao Tong University |
| NCT06739265 | Phase 1/Phase 2 (Phase 2) | Sep 1, 2024 | Chinese Academy of Medical Sciences |
| NCT06573138 | Phase 2 | Sep 1, 2024 | Jiao Tong University |
| NCT07234162 | Phase 3 | May 13, 2024 | Dizal (Jiangsu) Pharmaceutical Co., Ltd., Jiao Tong University |
Showing 20 of 22 trials
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Organizations
Research & Development (10)
| Organization | Org type | Trials | As lead sponsor | Phases | Earliest year |
|---|---|---|---|---|---|
| Jiao Tong University | Academic/Hospital | 7 | 6 | 2 | 2024 |
| Sun Yat-Sen University | Academic/Hospital | 4 | 4 | 1 | 2024 |
| Chinese Academy of Medical Sciences | Academic/Hospital | 3 | 3 | 1 | 2024 |
| Dizal (Jiangsu) Pharmaceutical Co., Ltd. | For profit | 3 | 1 | 2 | 2024 |
| Peking University | Academic/Hospital | 3 | 3 | 2 | 2024 |
| China Academy of Chinese Medical Sciences | Academic/Hospital | 1 | 1 | 1 | 2025 |
| Fudan University | Academic/Hospital | 1 | 1 | 1 | 2025 |
| Guangzhou Medical University | Academic/Hospital | 1 | 1 | 1 | 2026 |
| Henan Medical University | Academic/Hospital | 1 | 1 | 1 | 2023 |
| University of Texas at Houston | Academic/Hospital | 1 | 1 | 1 | 2025 |
10 organizations
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