← Mechanisms of action

JAK1

SINGLE PROTEINRattus norvegicus
Preferred name: Jak1 protein ChEMBL ↗

Linked proteins

Drugs acting on this target (30)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
abrocitinib (Cibinqo)AntagonistapprovedSmall moleculeJAK1 antagonist
arq-252InhibitorexperimentalSmall moleculeJAK1 inhibitor
ati-1777InhibitorexperimentalSmall moleculeJAK1 inhibitor
azd0449InhibitorexperimentalSmall moleculeJAK1 inhibitor
azd4205InhibitorexperimentalSmall moleculeJAK1 inhibitor
azd4604InhibitorexperimentalSmall moleculeJAK1 inhibitor
cee321InhibitorexperimentalSmall moleculeJAK1 inhibitor
cj-15314InhibitorexperimentalSmall moleculeJAK1 inhibitor
elsubrutinibInhibitorexperimentalSmall moleculeJAK1 inhibitor
fzj-003InhibitorexperimentalSmall moleculeJAK1 inhibitor
glpg3121InhibitorexperimentalSmall moleculeJAK1 inhibitor
golidocitinibInhibitorexperimentalSmall moleculeJAK1 inhibitor
IfidancitinibInhibitorexperimentalSmall moleculeJAK1 inhibitor
jacketinibInhibitorexperimentalSmall moleculeJAK1 inhibitor
kl130008InhibitorexperimentalSmall moleculeJAK1 inhibitor
leo 142397InhibitorexperimentalSmall moleculeJAK1 inhibitor
LorpucitinibInhibitorexperimentalSmall moleculeJAK1 inhibitor
max-40070InhibitorexperimentalSmall moleculeJAK1 inhibitor
pf06263276InhibitorexperimentalSmall moleculeJAK1 inhibitor
qy201InhibitorexperimentalSmall moleculeJAK1 inhibitor
qy211InhibitorexperimentalSmall moleculeJAK1 inhibitor
td-0903InhibitorexperimentalSmall moleculeJAK1 inhibitor
td-3504InhibitorexperimentalSmall moleculeJAK1 inhibitor
td-8236InhibitorexperimentalSmall moleculeJAK1 inhibitor
tdm-180935InhibitorexperimentalSmall moleculeJAK1 inhibitor
tll018InhibitorexperimentalSmall moleculeJAK1 inhibitor
tofacitinib (xeljanz)InhibitorapprovedSmall moleculeJAK1 inhibitor
tq05105InhibitorexperimentalSmall moleculeJAK1 inhibitor
vc005InhibitorexperimentalSmall moleculeJAK1 inhibitor
vvn461InhibitorexperimentalSmall moleculeJAK1 inhibitor