tetrazepam

Small moleculeexperimental

Tetrazepam is a benzodiazepine derivative with anticonvulsant, anxiolytic, muscle relaxant and slightly hypnotic properties. It was formerly used mainly in Austria, France, Belgium, Germany and Spain to treat muscle spasm, anxiety disorders such as panic attacks, or more rarely to treat depression, premenstrual syndrome or agoraphobia. Tetrazepam has relatively little sedative effect at low doses while still producing useful muscle relaxation and anxiety relief. The Co-ordination Group for Mutual Recognition and Decentralised Procedures-Human endorsed the Pharmacovigilance Risk Assessment Committee (PRAC) recommendation to suspend the marketing authorisations of tetrazepam-containing medicines across the European Union (EU) in April 2013. The European Commission has confirmed the suspension of the marketing authorisations for Tetrazepam in Europe because of cutaneous toxicity, effective from the 1 August 2013. — Wikipedia

Clinical trial activity

0 trials · 0 clinical orgs · 0 marketing orgs

Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0

Mechanism of action

Chemistry & pharmacology

Loading structure…

SMILES

CN1C(=O)CN=C(C2=CCCCC2)c2cc(Cl)ccc21
Mol. weight
288.78 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Achiral Molecule
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • 1a brand of tetrazepam
  • 4621 cb
  • 7-chloro-5-(1-cyclohexen-1- yl)-1,3-dihydro-1-methyl-2h-1,4-benzodiazepin-2-one
  • abz brand of tetrazepam
  • cb-4261
  • cb-4261
  • ct-arzneimittel brand of tetrazepam
  • fornet brand of tetrazepam
  • gry brand of tetrazepam
  • hexal brand of tetrazepam
  • krewel brand of tetrazepam
  • lichtenstein brand of tetrazepam
  • merck dura brand of tetrazepam
  • mibe brand of tetrazepam
  • mip brand of tetrazepam
  • mobiforton
  • mtw brand of tetrazepam
  • mtw-tetrazepam
  • musapam
  • musaril
  • myolastan
  • myolastan
  • myospasmal
  • panos
  • rilex
  • sanofi synthelabo brand of tetrazepam
  • tad brand of tetrazepam
  • tethexal
  • tetramdura
  • tetrarelax
  • tetra-saar
  • tetrazep 1a pharma
  • tetrazep abz
  • tetrazepam
  • tetrazepam
  • tetrazepam
  • tetrazepam
  • tetrazepam
  • tetrazepam
  • tetrazepam
  • tetrazep von ct