lypressin

Trade name: diapid

Small moleculeapproved

Lypressin is synthetic analog of porcine antidiuretic hormone vasopressin. Itis a cyclic nonapeptide that differs from Arg-vasopressin by one amino acid, containing Lys at residue 8 instead of Arg. Lypressin-containing nasal spray was used to treat diabetes insipidus, but its marketing by Sandoz (Novartis) was discontinued. — NCATS

Clinical trial activity

0 trials · 0 clinical orgs · 2 marketing orgs

Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0

Timeline

1960s

  1. Jul 11, 1967

    Sandoz — First NDA Organization

  2. Jul 11, 1967

    Sandoz — NDA Organization

Indications

Approved for

Mechanism of action

Approval history

  • approved

Chemistry & pharmacology

Loading structure…

SMILES

NCCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CSSC[C@H](N)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N1)C(=O)NCC(N)=O
Mol. weight
1056.24 g/mol
Chirality
Single Stereoisomer
Inorganic
No
Polymer
No
Delivery
Topical
Availability
Discontinued

Oral

No

Parenteral

No

Topical

Yes

Sources

Also known as

  • diapid
  • diapid
  • diapid
  • l-8
  • l-8
  • lypressin
  • lypressin
  • lypressin
  • lypressin
  • lypressin
  • lypressin
  • lypressin
  • lypressin
  • lypressin
  • lysine pitressin
  • lysine vasopressin
  • lysipressin
  • lysopressin
  • lysylvasopressin
  • syntopressin

Organizations

Marketing (2)

OrganizationOrg typeRelationshipDate
NovartisFor profitNDA2
SandozFor profitNDAJul 11, 1967