CDEK
← Mechanisms of action

AVPR1A

SINGLE PROTEINHomo sapiens
Preferred name: Vasopressin V1a receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (15)

Active Pharmaceutical Ingredient Mechanism Type ▲ Approval Status API Type Mechanism of Action
FelypressinActivatorexperimentalSmall moleculeAVPR1A activator
phin-214AgonistexperimentalSmall moleculeAVPR1A agonist
selepressinAgonistexperimentalSmall moleculeAVPR1A agonist
vasopressin (vasostrict)AgonistapprovedAnimal productAVPR1A agonist
balovaptanAntagonistexperimentalSmall moleculeVasopressin V1a receptor antagonist
bay 1753011AntagonistexperimentalSmall moleculeAVPR1A antagonist
conivaptan (vaprisol)AntagonistapprovedSmall moleculeAVPR1A antagonist
nmra-323511AntagonistexperimentalSmall moleculeAVPR1A antagonist
relcovaptanAntagonistexperimentalSmall moleculeAVPR1A antagonist
ro5285119AntagonistexperimentalSmall moleculeAVPR1A antagonist
srx-246AntagonistexperimentalSmall moleculeAVPR1A antagonist
srx-251AntagonistexperimentalSmall moleculeAVPR1A antagonist
va111913AntagonistexperimentalSmall moleculeAVPR1A antagonist
balovaptanInhibitorexperimentalSmall moleculeAVPR1A inhibitor
oce-205Partial agonistexperimentalSmall moleculeAVPR1A partial agonist