← Mechanisms of action
DNA polymerase (alpha/delta/epsilon)
PROTEIN FAMILYHomo sapiens
Linked proteins
- DNA polymerase alpha catalytic subunit (POLA1) ↗
- DNA polymerase delta subunit 4 (POLD4) ↗
- DNA polymerase delta subunit 3 (POLD3) ↗
- DNA polymerase delta catalytic subunit (POLD1) ↗
- DNA polymerase delta subunit 2 (POLD2) ↗
- DNA polymerase epsilon catalytic subunit A (POLE) ↗
- DNA polymerase alpha subunit B (POLA2) ↗
- DNA primase small subunit (PRIM1) ↗
- DNA primase large subunit (PRIM2) ↗
- DNA polymerase epsilon subunit 2 (POLE2) ↗
- DNA polymerase epsilon subunit 3 (POLE3) ↗
Drugs acting on this target (6)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| Aspacytarabine | Inhibitor | experimental | Small molecule | DNA polymerase (alpha/delta/epsilon) inhibitor |
| clofarabine (clolar) | Inhibitor | approved | Small molecule | DNA polymerase (alpha/delta/epsilon) inhibitor |
| cytarabine (cytosar-u) | Inhibitor | approved | Small molecule | DNA polymerase (alpha/delta/epsilon) inhibitor |
| fludarabine (fludara) | Inhibitor | approved | Small molecule | DNA polymerase (alpha/delta/epsilon) inhibitor |
| gemcitabine (gemzar) | Inhibitor | approved | Small molecule | DNA polymerase (alpha/delta/epsilon) inhibitor |
| troxatyl | Inhibitor | experimental | Small molecule | DNA polymerase (alpha/delta/epsilon) inhibitor |