← Mechanisms of action

HTR1B

SINGLE PROTEINHomo sapiens
Preferred name: Serotonin 1b (5-HT1b) receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (15)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
almotriptan (axert)AgonistapprovedSmall moleculeHTR1B agonist
donitriptanAgonistexperimentalSmall moleculeHTR1B agonist
eletriptan (relpax)AgonistapprovedSmall moleculeHTR1B agonist
eltoprazineAgonistexperimentalSmall moleculeHTR1B agonist
ergoloid mesylateAgonistapprovedSmall moleculeHTR1B agonist
frovatriptan (frova)AgonistapprovedSmall moleculeHTR1B agonist
MethylergonovineAgonistexperimentalBiologicalHTR1B agonist
naratriptan (amerge)AgonistapprovedSmall moleculeHTR1B agonist
rizatriptan (maxalt)AgonistapprovedSmall moleculeHTR1B agonist
sumatriptan (zecuity)AgonistapprovedSmall moleculeHTR1B agonist
t521AgonistexperimentalAllergenHTR1B agonist
zolmitriptan (zomig)AgonistapprovedSmall moleculeHTR1B agonist
gsk163090AntagonistexperimentalSmall moleculeHTR1B antagonist
trelanserinAntagonistexperimentalSmall moleculeHTR1B antagonist
xc130-a10hAntagonistexperimentalSmall moleculeHTR1B antagonist